Theliatinib

CAS NO.:1353644-70-8

Molecular Formula:C₂₅H₂₆N₆O₂

Molecular Weight:442.51

Purity: > 98%

Solubility (R.T.: 25℃): DMSO

Stability: - 20℃ 2 years

Theliatinib (HMPL-309) is a potent, ATP-competitive, orally active and highly selective EGFR inhibitor with a Ki of 0.05 nM and an IC50 of 3 nM.Theliatinib has an IC50 of 22 nM for EGFR T790M/L858R mutant.Theliatinib shows >50-fold selectivity for EGFR th

We offer significant discount for larger quantity order.

For quotation, question, and order, please send email to sales@rechemscience.com

Quality Control by H-NMR,C-NMR,LC-MS,HPLC.

Product will be shipped with supporting analytical data.

Fast delivery about 4-5 working days.