| R1133388 |
MSC-4381 |
MSC-4381 (MCT4-IN-1), a chemical probe, is an orally active and selective monoca
|
| R1133389 |
Zerencotrep |
Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels, inhibits (-)-e
|
| R1133390 |
Wnt pathway activator 2 |
Wnt pathway activator 2 (compound 2) is a potent Wnt activator with an EC50 of 1
|
| R1133391 |
8-OH-DPAT hydrobromide |
8-OH-DPAT (8-Hydroxy-DPAT) hydrobromide is a potent, brain-penetrant and selecti
|
| R1133392 |
STAT3-IN-3 |
STAT3-IN-3 is a potent and selective inhibitor of signal transducer and activato
|
| R1133393 |
Rocbrutinib |
Rocbrutinib is an orally available, highly selective Bruton's tyrosine kinase (B
|
| R1133394 |
RBN012759 |
RBN012759 is a potent, selective and orally active inhibitor of PARP14, with an
|
| R1133397 |
DDO-5936 |
DDO-5936 is a potent and specific Hsp90-Cdc37 PPI inhibitor.
|
| R1133398 |
KU-0060648 |
KU-0060648 is a dual inhibitor of PI3K and DNA-PK with IC50s of 4 nM, 0.5 nM, 0.
|
| R1133399 |
Dasminapant(APG-1387) |
Dasminapant (APG-1387), a bivalent SMAC mimetic and an IAP antagonist, blocks th
|
| R1133400 |
PFI-2 hydrochloride |
PFI-2 hydrochloride ((R)-PFI-2 hydrochloride) is a potent, highly selective, and
|
| R1133401 |
PFI-2 |
PFI-2 is an effective, specific and cell-active lysine methyltransferase SETD7 i
|
| R11335103 |
GGFG-PAB-Exatecan |
GGFG-PAB-Exatecan consists of an ADC toxin Exatecan (HY-13631) and a linker GGFG
|
| R1133402 |
Droperidol |
Droperidol (Dehydrobenzperidol) is a butyrophenone pamine-2 receptor antagonist
|
| R1133403 |
SG-094 |
SG-094 is a potent TPC2 inhibitor with antiproliferative effects.
|
| R1133404 |
ARV-471 |
Vepdegestrant (ARV-471) is an orally active PROTAC estrogen receptor degrader.
|
| R1133405 |
HIV-1 inhibitor-69 |
HIV-1 inhibitor-69 is an HIV-1 reverse transcriptase inhibitor.
|
| R1133406 |
SB-215505 |
SB-215505 is an orally active and subtype-selective 5-HT2B receptor antagonist w
|
| R1133407 |
JS11 |
JS11 is an inhibitor for natriuretic polypeptide receptor 1 (Npr1) with an IC50
|
| R1133408 |
Carboxyamidotriazole |
Carboxyamidotriazole (L-651582) is an orally active cytostatic inhibitor of nonv
|
| R1133409 |
LY 311727 |
LY-311727 is a potent secretory non-pancreatic phospholipase A2 (sPLA2) inhibito
|
| R1133410 |
Vopimetostat(TNG-462) |
TNG-462 is an orally active and selective PRMT5 inhibitor.
|
| R1133411 |
GNE-495 |
GNE-495 is a potent and selective MAP4K4 inhibitor with an IC50 of 3.7 nM.
|
| R1133412 |
NIBR-17 |
NIBR-17 is a pan-class I PI3K inhibitor with suitable pharmacokinetic properties
|
| R1133413 |
L-372662 |
L-372662 is a potent and orally active non-peptide oxytocin antagonist with a Ki
|