R2032333 |
ABT-346 |
ATB-346 is a novel hydrogen sulphide-releasing derivative of naproxen with marke
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R2032334 |
ABT-751(E7010) |
ABT-751(E 7010) is a novel bioavailable tubulin-binding and antimitotic sulfonam
|
R2032335 |
AdipoRon |
AdipoRon is an orally active adiponectin receptor (AdipoR) agonist, binding to A
|
R2032336 |
ADL5859 |
ADL5859 is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against op
|
R2032337 |
AG1024(Tyrphostin AG 1024) |
AG1024 (Tyrphostin AG 1024) is a reversible, competitive and selective insulin-l
|
R2032338 |
AM251 |
AM251 is a selective cannabinoid 1 (CB1) receptor antagonist with an IC50 of 8 n
|
R2032339 |
AM-281;AM281 |
Potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values
|
R2032340 |
AMG837 |
AMG 837 is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic pr
|
R2032341 |
AMG900 |
AMG 900 is a potent and highly selective pan-Aurora kinases inhibitor with IC50
|
R2032342 |
AT13148 |
AT13148 is an orally active and ATP-competitive, multi-AGC kinase inhibitor with
|
R2032343 |
AT-7867 |
AT7867 is a potent ATP-competitive inhibitor of Akt1/Akt2/Akt3 and p70S6K/PKA wi
|
R2032344 |
Avelestat(AZD9668) |
Alvelestat (AZD9668) is an orally bioavailable, affinity and selective inhibitor
|
R2032345 |
AVP-AEW541;AEW541 |
NVP-AEW541 is a potent inhibitor of IGF-1R with IC50 of 0.15 μM, also inhibits I
|
R2032346 |
AZ191 |
AZ191 is a potent inhibitor that selectively inhibits DYRK1B with IC50 of 17 nM.
|
R2032347 |
AZ20 |
AZ20 is a potent and selective inhibitor of ATR with an IC50 of 5 nM, and has 8-
|
R2032348 |
AZ3146 |
AZ3146 is a reasonably potent and selective Mps1 inhibitor with IC50 of 35 nM fo
|
R2032349 |
AZ960 |
AZ960 is a potent and specific inhibitor of the JAK2 kinase with a Ki of 0.45 nM
|
R2032350 |
Barasertib-HQPA;AZD2811;INH-34;AZD1152-HQPA |
Barasertib-HQPA (AZD2811) is a highly selective Aurora B inhibitor with an IC50
|
R2032351 |
AZD1208 |
AZD1208 is a novel, orally bioavailable, highly selective PIM kinases inhibitor.
|
R2032352 |
AZD1283 |
AZD1283 is a potent antagonist of the P2Y12 receptor with EC50 of 3.0 ug/kg/min,
|
R2032353 |
Vistusertib (AZD2014) |
Vistusertib (AZD2014) is an ATP competitive mTOR inhibitor with an IC50 of 2.81
|
R2032354 |
AZD2932 |
AZD2932 is a potent and multi-targeted kinase inhibitor VEGFR2, PDGFβ, Flt-3 and
|
R2032355 |
AZD3514 |
AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM a
|
R2032356 |
AZD6482;AZD 6482 (KIN-193) |
AZD 6482 (KIN-193) is a potent and selective p110β inhibitor with an IC50 of 0.6
|
R2032357 |
AZD7545 |
AZD7545 is a potent, competitive, selective PDHK2 (pyruvate dehydrogenase kinase
|