R2032383 |
Fimepinostat(CUDC-907) |
Fimepinostat (CUDC-907) potently inhibits class I PI3Ks as well as classes I and
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R2032384 |
CX5461 |
CX-5461 is a potent and oral rRNA synthesis inhibitor.It inhibits RNA polymerase
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R2032385 |
CX-6258 |
CX-6258 is a potent and kinase selective pan-Pim kinases inhibitor, with IC50s o
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R2032386 |
CZC24832 |
CZC24832 is a highly selective and potent PI3Kγ inhibitor (IC50=27 nM) with appa
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R2032387 |
Dalcetrapib(JTT-705;RO4607381) |
Dalcetrapib (JTT-705; RO-4607381) is a rhCETP inhibitor with IC50 of 0.2 μM that
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R2032388 |
Dasabuvir(ABT-333) |
Dasabuvir (ABT-333) is a nonnucleoside inhibitor of the RNA-dependent RNA polyme
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R2032389 |
DCC-2036(Rebastinib) |
Rebastinib (DCC-2036) is a conformational control Bcr-Abl inhibitor for Abl1WT a
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R2032390 |
c-Kit-IN-1 |
c-Kit-IN-1 is a potent inhibitor of c-Kit and c-Met with IC50s of <200 nM.
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R2032391 |
Degrasyn(WP1130) |
Degrasyn (WP1130) is a cell-permeable deubiquitinase (DUB) inhibitor, directly i
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R2032392 |
ELN441958 |
ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding
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R2032393 |
ENMD-2076 |
ENMD-2076 is a multi-targeted kinase inhibitor with IC50s of 1.86, 14, 58.2, 15.
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R2032394 |
EPZ004777 |
EPZ004777 is a potent, selective DOT1L inhibitor with an IC50 of 0.4 nM.
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R2032395 |
EPZ005687 |
EPZ005687 is a potent and selective inhibitor of EZH2 with Ki of 24 nM, and has
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R2032396 |
Pinometostat(EPZ-5676) |
Pinometostat (EPZ-5676) is a potent DOT1L histone methyltransferase inhibitor wi
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R2032397 |
ETP46464 |
ETP-46464 is an effective mTOR and ATR inhibitor with IC50s of 0.6 and 14 nM, re
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R2032398 |
FR 180204 |
FR 180204 is an ATP-competitive and selective ERK inhibitor.FR 180204 inhibits E
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R2032399 |
GNE-0877 |
GNE0877 is a highly potent, selective, and brain-penetrant aminopyrazole leucine
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R2032400 |
GNE-477 |
GNE-477 is a potent and efficacious dual PI3K (IC50=4 nM)/mTOR(Ki=21 nM) inhibit
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R2032401 |
GNE7915 |
GNE-7915 is a potent, selective and brain-penetrant inhibitor of LRRK2 with an I
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R2032402 |
GNE9605 |
GNE-9605 is a highly potent, selective, and brain-penetrant LRRK2 inhibitor with
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R2032403 |
GNF-5 |
GNF-5, an analogue of GNF-2 with improved pharmacokinetic properties, is a selec
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R2032404 |
GNF5837 |
GNF-5837 is a potent, selective, and orally bioavailable pan-tropomyosin recepto
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R2032405 |
GSK1292263 |
GSK1292263 is a novel GPR119 receptor agonist used for the treatment of type 2 d
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R2032406 |
GSK1904529A |
GSK1904529A is a selective inhibitor of IGF-1R and IR with IC50 of 27 nM and 25
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R2032407 |
GSK2334470 |
GSK2334470 is a highly specific and potent inhibitor of PDK1 with an IC50 of 10
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