R2033099 |
SM16 |
SM 16 is a ALK5/ALK4 kinase inhibitor with Kis of 10 and 1.5 nM, respectively.
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R2033100 |
Sotrastaurin |
Sotrastaurin is a potent and orally-active pan-PKC inhibitor, with Kis of 0.22 n
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R2033101 |
SP-13786 |
SP-13786 is a highly potent and selective inhibitor of fibroblast activation pro
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R2033102 |
SPHINX31 |
SPHINX31 is a potent and selective inhibitor of serine/arginine-rich protein kin
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R2033103 |
SR3677 |
SR-3677 is a potent and selective ROCK-II inhibitor with an IC50 of ~3 nM.
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R2033104 |
1358099-18-9 |
C25-140, a first-in-class, fairly selective TRAF6-Ubc13 inhibitor, directly bind
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R2033105 |
ACY775 |
ACY-775 is a potent and selective inhibitor of the of histone deacetylase 6 (HDA
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R2033106 |
Adavivint(SM04690;Lorecivivint) |
Adavivint (SM04690; Lorecivivint) is a potent and selective inhibitor of canonic
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R2033107 |
AR231453 |
AR 231453 is a potent, selective and orally available GPR119 agonist.
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R2033108 |
Asapiprant |
Asapiprant is a potent and selective DP1 receptor antagonist with a Ki of 0.44 n
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R2033109 |
AVN492 |
AVN-492 is a very specific and highly-selective antagonist with picomolar affini
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R2033110 |
AZ304 |
AZ304 is an ATP-competitive dual BRAF kinase inhibitor, potently inhibits wild t
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R2033111 |
AZD1390 |
AZD1390 is a potent, highly selective, orally bioavailable, brain-penetrant ATM
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R2033112 |
AZD5069 |
AZD-5069 is a potent CXCR2 chemokine receptor antagonist, used for caner treatme
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R2033113 |
BIBF1202 |
BIBF 1202 is the carboxylate metabolite of BIBF 1120 which inhibits VEGFR2 kinas
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R2033114 |
Desidustat |
Desidustat is an inhibitor of HIF hydroxylase extracted from patent WO 201410281
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R2033115 |
GNE-6776 |
GNE-6776 is a selective USP7 inhibitor.
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R2033116 |
GSK3179106 |
GSK3179106 is a potent and selective RET kinase inhibitor with an IC50 of 0.4 nM
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R2033117 |
Imepitoin |
Imepitoin (AWD 131-138) is a new low-affinity partial benzodiazepine receptor ag
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R2033118 |
JAK3-IN-6 |
JAK3-IN-6 is a potent, selective irreversible Janus Associated Kinase 3 (JAK3) i
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R2033119 |
LY-2940094 tartrate |
LY-2940094 is a potent, selective and orally available nociceptin receptor (NOP
|
R2033120 |
LY-2940094;LY2940094 |
LY-2940094 is a potent, selective and orally available nociceptin receptor (NOP
|
R2033121 |
LY3023414 |
LY3023414 potently and selectively inhibits class I PI3K isoforms, DNA-PK, and m
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R2033122 |
Nec-1s |
Necrostatin 2 racemate (Nec-1S), the Nec-1 stable, is a potent and specific RIPK
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R2033123 |
Nucleozin |
Nucleozin targets influenza A nucleoprotein (NP), a multifunctional, RNA-binding
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