R2101233 |
acivicin;AT-125; U-42126 |
Acivicin (AT-125), a natural product produced by Streptomyces sviceus, is a γ−gl
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R2101234 |
Cenicriviroc(mesylate) |
Cenicriviroc Mesylate is a dual CCR2/CCR5 antagonist, also inhibits both HIV-1 a
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R2101235 |
AZD4573 |
AZD4573 is an effective and selective CDK9 inhibitor (IC50: <4 nM). It enable
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R2101236 |
WYE-354 |
WYE-354(IC50=5 nM) is an effective, selective and ATP-competitive mTOR inhibitor
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R2101237 |
ML-SA1 |
activator of TRPML channels.
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R2101238 |
Fezolinetant |
Fezolinetant is an antagonist of the neurokinin 3 receptor (NK3R). It is used fo
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R2101239 |
AZD-4320 |
AZD4320 is an inhibitor of BH3-mimicking dual BCL2/BCLxL. For KPUM-MS3, KPUM-UH1
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R2101240 |
RTA 405 |
CDDO-EA is an activator of NF-E2 related factor 2/antioxidant response element (
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R2101241 |
BDTX-189 |
BDTX-189 is an orally bioavailable, irreversible, selective, small-molecule inhi
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R2101242 |
E3 Ligase Ligand-Linker Conjugates 2 |
E3 Ligase Ligand-Linker Conjugates 2 is a synthesized E3 ligase ligand-linker co
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R2101243 |
E3 ligase Ligand-Linker Conjugates 28 |
(S,R,S)-AHPC-C4-NH2 hydrochloride is a synthesized E3 ligase ligand-linker conju
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R2101244 |
E3 Ligase Ligand-Linker Conjugates 20 |
Thalidomide-O-amido-C8-NH2 (Cereblon Ligand-Linker Conjugates 2), a synthesized
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R2101245 |
E3 ligase Ligand-Linker Conjugates 7 |
(S,R,S)-AHPC-PEG4-NH2 hydrochloride is a synthesized E3 ligase ligand-linker con
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R2101246 |
BSJ-03-123 |
BSJ-03-123 is a Selective Cdk6 degrader. BSJ-03-123 exploits protein-interface d
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R2101247 |
VH032-C10-NH2 dihydrochloride |
(S,R,S)-AHPC-C10-NH2 dihydrochloride (VH032-C10-NH2 dihydrochloride) is a synthe
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R2101248 |
VH032-C4-NH2 |
(S,R,S)-AHPC-C4-NH2 is a synthesized E3 ligase ligand-linker conjugate that inco
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R2101249 |
AT1 |
BRD4 degrader AT1 is a highly selective Brd4 degrader based on PROTAC technology
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R2101250 |
dBET57 |
dBET57 is heterobifunctional degrader of BRD4 based on the PROTAC technology, ex
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R2101251 |
(S)-AZD6738 |
(S)-Ceralasertib is a potent and selective inhibitor of sulfoximine morpholinopy
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R2101252 |
MS4078 |
MS4078 is an anaplastic lymphoma kinase (ALK) PROTAC. It has a Kd of 19 nM for b
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R2101253 |
(S)-JQ-35 |
(S)-JQ-35 (TEN-010) is an inhibitor of the Bromodomain and Extra-Terminal (BET)
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R2101254 |
A1874 |
A1874 is a nutlin-based and BRD4-degrading PROTAC which induces BRD4 degradation
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R2101255 |
TL13-112 |
TL13-112 is a selective degrader of ALK-PROTAC and inhibits ALK activity (IC50:
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R2101256 |
CCT367766 |
CCT367766 is the PROTAC-based pirin targeting protein degradation probe, deplete
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R2101258 |
MS1943 |
MS1943 is a orally bioavailable EZH2 selective degrader(IC50 of 120 nM).
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