R21082415 |
SGC-GAK-1 |
Sgc-gak-1 is a potent selective cyclin G-associated kinase (GAK) inhibitor with
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R21082416 |
S-GBOXIN |
S-gboxin is an active analogue of Gboxin and has potent antitumor activity.
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R21082417 |
Voxelotor |
GBT 440 (Voxelotor) is an orally available regulator of sickle cell hemoglobin.
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R21082418 |
NSC23766 3HCL |
NSC 23766 trihydrochloride is an inhibitor of Rac1 activation.
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R21082419 |
IC-87201 |
IC87201 is an inhibitor of psD95-NNOS interaction, which inhibits the formation
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R21082420 |
AMG837 (calcium hydrate) |
AMG 837 calcium hydroxide is a GPR40 agonist with EC50 of 13 nM and has good pha
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R21082421 |
CAY10650 |
CAY10650 is a cPLA2α inhibitor with IC50 of 12 nM.
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R21082422 |
DKM2-93 |
DKM 2-93 is a relatively selective inhibitor of UBA5 with IC50 value of 430 μM.
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R21082423 |
PF429242 dihydrochloride |
PF429242 dihydrochloride is a reversible and competitive inhibitor of S1P (IC50
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R21082424 |
AZ1 |
USP25/28 inhibitor AZ1 (AZ1) is a potent, selective, and non-competitive dual ub
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R21082425 |
MB-07811 ( VK-2809) |
Mb-07811 (VK-2809) is a HepDirect prodrug with oral activity of MB07344, a liver
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R21082426 |
Udenafil |
Udenafil(DA8159) is a PDE5 inhibitor.
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R21082427 |
RHC-80267 |
RHC 80267 (U-57908) is an effective selective diacylglycerase (DAGL) inhibitor (
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R21082428 |
JWG-071 |
Jwg-071 is the first reported ERK5 kinase selective chemical probe. Jwg-071 imp
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R21082429 |
RIPASUDIL |
Ripasudil Free Base (K-115 Free Base) is a rock-specific inhibitor that inhibits
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R21082430 |
JDTIC |
JDTic is a κ- opioid receptor antagonist, but has no effect on μ- and δ- opioid
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R21082431 |
Dual Specificity Protein Phosphatase 1/6 Inhibitor |
(E/Z)-BCI (NSC 150117) is a DUSP6 inhibitor with anti-inflammatory activity. (E
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R21082432 |
VAS2870 |
VAS2870 is NADPH oxidase (NOX) inhibitor.
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R21082433 |
Nelonicline |
Nelonicline (ABT-126) is a selective agonist of neuronal nicotinic receptors.
|
R21082434 |
VBIT-12 |
Vbit-12 is a potent inhibitor of VDAC1. Vbit-12 interacts directly with VDAC1 a
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R21082435 |
SR-18292 |
Sr-18292 is an inhibitor of PPARγ co-activator -1α (PGC-1α), which promotes the
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R21082436 |
Belvarafenib |
Belvarafenib is an effective, widespread rapidly accelerating fibrosarcoma kinas
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R21082437 |
Ingliforib |
Ingliforib is a glycogen phosphorylase inhibitor with IC50 values of 52,352 nM a
|
R21082438 |
GSK3117391A |
Dac-in-3 is an inhibitor of histone deacetylase (HDAC). For details, please refe
|
R21082439 |
Vindesine |
The semi-synthetic vinblastine derivatives have higher anti-cancer spectrum, hig
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