R2032879 |
MK8931;Verubecestat(MK-8931) |
Verubecestat (MK-8931) is a beta-secretase 1 (BACE1) inhibitor under investigati
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R2032880 |
PI-1840 |
PI-1840 is a potent and selective inhibitor for chymotrypsin-like (CT-L) (IC50 v
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R2032881 |
PNU74654 |
PNU-74654 is an inhibitor of Wnt/β-catenin pathway with an IC50 of 129.8 μM in N
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R2032882 |
RAD-140 |
RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen recepto
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R2032883 |
Rbin-1 |
Rbin-1 is a potent, reversible, and specific chemical inhibitor of eukaryotic ri
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R2032884 |
SAR405 |
SAR405 is a first-in-class, selective, and ATP-competitive PI3K class III (PIK3C
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R2032885 |
VER49009 |
VER-49009 is a Hsp90 inhibitor, with an IC50 of 25 nM and a Kd of 78 nM.
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R2032886 |
VER50589 |
VER-50589 is a Hsp90 inhibitor, with an IC50 of 21 nM and a Kd of 4.5 nM.
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R2032887 |
AMG9810 |
AMG9810 is a selective and competitive vanilloid receptor 1 (TRPV1) antagonist w
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R2032888 |
TGR1202 |
Umbralisib (TGR-1202) is a novel PI3Kδ inhibitor, with IC50 and EC50 of 22.2 nM
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R2032889 |
Cenicriviroc |
Cenicriviroc is an orally active, dual CCR2/CCR5 antagonist, also inhibits both
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R2032890 |
DiZPK |
DiZPK is a photocrosslinker for identifying direct protein-protein interactions
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R2032891 |
EED226 |
EED226 is a polycomb repressive complex 2 (PRC2) inhibitor, which binds to the K
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R2032892 |
GLPG0187 |
GLPG0187 is a broad spectrum integrin receptor antagonist with antitumor activit
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R2032893 |
ML385 |
ML385 is a specific nuclear factor erythroid 2-related factor 2 (NRF2) inhibitor
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R2032894 |
PF-06282999 |
PF-06282999 is a potent and selective myeloperoxidase inhibitor which is potenti
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R2032895 |
WT-161 |
WT-161 is a potent and selective HDAC6 inhibitor with an IC50 of 0.40 nM.
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R2032896 |
AP-III-a4 |
ENOblock(AP-III-a4) is a novel small molecule which is the first, nonsubstrate a
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R2032897 |
ARN272 |
ARN272 is an anandamide transport inhibitor.
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R2032898 |
AS1842856 |
AS1842856, a specific Foxo1 inhibitor (IC50=30 nM), potently suppresses autophag
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R2032899 |
BIBS39 |
BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist.Target: Ang
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R2032900 |
CCT245737 |
CCT245737 is an orally active and seletive Chk1 inhibitor, with an IC50 of 1.3 n
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R2032901 |
Grapiprant |
Grapiprant (CJ-023423) is a selective EP4 receptor antagonist whose physiologica
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R2032902 |
HG-14-10-04 |
HG-14-10-04 is a potent and specific ALK inhibitor with IC50 of 20 nM.IC50 value
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R2032903 |
WNK463 |
WNK463 is an orally bioavailable pan-With-No-Lysine (K) (WNK)-kinase inhibitor w
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