R2101146 |
SAR-020106 |
SAR-020106 is an ATP-competitive, potent, and selective CHK1 inhibitor with an I
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R2101147 |
A-893 |
A-893 is a cell-active inhibitor of Methyltransferase SMYD2, with an IC50 of 2.8
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R2101148 |
Mirogabalin besylate |
Mirogabalin besylate is a selective and orally available ligand for the α2δ subu
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R2101149 |
Px-104 |
(-)-PX20606 trans isomer is an agonist of FXR (EC50s: 18 and 29 nM for FXR in FR
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R2101150 |
RUC-4 |
RUC-4 (RUC4;RUC 4) is a potent, selective, non-RGD-mimetic αIIbβ3 integrin recep
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R2101151 |
GDC-0077 |
GDC-0077 (RG6114) is a potent, orally available, and selective inhibitor of PI3K
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R2101152 |
CYC065;CDK259 |
CYC065 is an orally available, second-generation ATP-competitive inhibitor of CD
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R2101153 |
LX-2761 |
LX2761 is a chemically stable and effective inhibitor against sodium-dependent g
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R2101154 |
Baloxavir |
Baloxavir is a first-in-class cap-dependent endonuclease inhibitor of the influe
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R2101155 |
ARS-1323 |
ARS-1323 (the racemate of ARS-1620) is a mutant K-ras G12C inhibitor extracted f
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R2101156 |
CDDO-2-P-Im |
CDDO-3P-Im, an analog of CDDO-Imidazolide, has a chemopreventive effect. It can
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R2101157 |
R-268712 |
R-268712 is an effective and selective inhibitor of ALK5 IC50: 2.5 nM).
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R2101158 |
BAZ2-ICR |
BAZ2-ICR is an epigenetic chemical probe and it also is a potent, selective, cel
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R2101159 |
QC6352 |
QC6352 is a selective and effective KDM4C inhibitor (IC50: 35 nM).
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R2101160 |
T-26c |
T-26c is highly potent and selective matrix metalloproteinase-13 (MMP-13) inhibi
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R2101161 |
CDDO-2-P-Im |
CDDO-2P-Im, an analog of CDDO-Imidazolide, has a chemopreventive effect. It can
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R2101162 |
TP 235 |
CDDO-Im is an activator of Nrf2 and PPAR (Kis: 232/344 nM for PPARα/PPARγ).
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R2101163 |
BAY 299 |
BAY-299 is a very potent inhibitor. For BRPF2 bromodomains (BD), TAF1 BD2, TAF1L
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R2101164 |
BMS-955176;GSK3532795 |
GSK3532795 is a potent, orally active, second-generation HIV-1 maturation inhib
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R2101165 |
Quarfloxin |
Quarfloxin is a fluoroquinolone derivative with antineoplastic activity with IC5
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R2101166 |
BI-3802 |
BI-3802 is a highly effective BCL6 depressant, which can inhibit the BTB domain
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R2101167 |
GSK-484 |
GSK484 is a potent PAD-4 inhibitor (Protein-arginine deiminase type-4). GSK484 p
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R2101168 |
BAY-850 |
BAY-850 is a potent and isoform selective ATPase family AAA domain-containing pr
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R2101169 |
SB-204990 |
SB 204990 is an effective and specific ATP citrate lyase enzyme inhibitor.
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R2101170 |
Quarfloxin |
Quarfloxin (CX 3543) 是一种具有抗肿瘤活性的氟喹诺酮类衍生物,其靶向抑制RNA pol I的活性,在神经母细胞瘤中的IC50 值在纳摩尔级别
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