R2032514 |
Rigosertib(ON-01910) |
Rigosertib (ON-01910) is a non-ATP-competitive inhibitor of PLK1 with IC50 of 9
|
R2032515 |
RKI-1447 |
RKI-1447 is a potent small molecule inhibitor of ROCK1 and ROCK2 with IC50 value
|
R2032516 |
RN486 |
RN486 is a selective Btk inhibitor with an IC50 Value of 4.0 nM.IC50 Value: 4.0
|
R2032517 |
RO5126766(CH5126766) |
Ro 5126766 is a first-in-class dual MEK/RAF inhibitor that allosterically inhibi
|
R2032518 |
SAL003 |
Sal003 is a potent, specific and cell-permeable inhibitor of the eukaryotic tran
|
R2032519 |
SB1317 Hydrochloride(TG02) |
SB1317 is a potent inhibitor of CDK2, JAK2, and FLT3 for the treatment of cancer
|
R2032520 |
SB271046 |
SB271046 Hcl is a potent, selective and orally active 5-HT6 receptor antagonist
|
R2032521 |
SB505124 |
SB-505124 is a selective inhibitor of TGF-β Receptor type I receptor (ALK4, ALK5
|
R2032522 |
SB743921 |
SB-743921 is a potent inhibitor of the mitotic kinesin KSP (Eg5), with a Ki of 0
|
R2032523 |
SC-514 |
SC-514 is a selective IKK-2 inhibitor (IC50=11.2±4.7 μM), which does not inhibit
|
R2032524 |
SGC0946 |
SGC0946 is a highly potent and selective DOT1L methyltransferase inhibitor with
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R2032525 |
SGX-523 |
SGX-523 is a selective Met inhibitor with IC50 of 4 nM, no activity to BRAFV599E
|
R2032526 |
Skepinone-L;CBS3830 |
Skepinone-L (CBS3830) is a selective p38 mitogen-activated protein kinase inhibi
|
R2032527 |
SKLB1002 |
SKLB1002 is a potent and ATP-competitive VEGFR2 inhibitor with IC50 of 32 nM.
|
R2032528 |
SKLB610 |
SKLB1002 is a potent and ATP-competitive VEGFR2 inhibitor with IC50 of 32 nM.
|
R2032529 |
SNS-032(BMS-387032) |
SNS-032 (BMS-387032) is a selective inhibitor of CDK2, CDK7, and CDK9 with IC50s
|
R2032530 |
SNS-314 Mesylate |
SNS-314 is a potent and selective aurora kinase inhibitor with IC50s of 9, 31, a
|
R2032531 |
SSR128129E |
SSR128129E is an orally available and allosteric FGFR inhibitor with an IC50 of
|
R2032532 |
SteMRegenin 1 |
StemRegenin 1 is a potent aryl hydrocarbon receptor (AhR) antagonist with IC50 o
|
R2032533 |
SU11274 |
SU11274 is a selective Met inhibitor with IC50 of 10 nM, but has no effects on P
|
R2032534 |
SU9516 |
SU9516 is a potent CDK2 inhibitor, with an IC50 of 22 nM, and also shows inhibit
|
R2032535 |
TAK-700(Orteronel) |
TAK-700 (Orteronel) is a potent and highly selective human 17,20-lyase inhibitor
|
R2032536 |
TAK733 |
TAK-733 is a potent and selective MEK allosteric site inhibitor with an IC50 of
|
R2032537 |
TAK875;Fasiglifam(TAK-875) |
Fasiglifam (TAK-875) is a selective GPR40 agonist with EC50 of 14 nM in human GP
|
R2032538 |
Talabostat Mesilate |
Talabostat mesylate (Val-boroPro mesylate; PT100 mesylate) is an orally active a
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