R2032591 |
PD184352;CI-1040 |
CI-1040 (PD 184352) is an orally active, highly specific, small-molecule inhibit
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R2032592 |
INCB39110 |
Itacitinib adipate is an orally bioavailable and selective JAK1 inhibitor which
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R2032593 |
SH-4-54 |
SH-4-54 is a most potent, small molecule, nonphosphorylated STAT inhibitor, with
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R2032594 |
UNC0638 |
UNC0638 selectively inhibits G9a and GLP histone methyltransferase activity with
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R2032595 |
ZSTK-474;ZSTK474 |
ZSTK474 is an ATP-competitive pan-class I PI3K inhibitor with IC50s of16 nM, 44
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R2032596 |
UNBS-5162;UNBS5162 |
UNBS5162 is a pan-antagonist of CXCL chemokine expression, with anti-tumor activ
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R2032597 |
FTI-277 hydrochloride |
FTI-277 hydrochloride is an inhibitor of farnesyl transferase (FTase); a highly
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R2032598 |
LY2090314 |
LY2090314 is a potent inhibitor of glycogen synthase kinase-3 (GSK-3) with IC50
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R2032599 |
ReModelin |
Remodelin hydrobromide is a novel potent and selective inhibitor of the acetyl-t
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R2032600 |
Ro48-8071 |
Ro 48-8071 fumarate is an inhibitor of OSC (Oxidosqualene cyclase) with IC50 of
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R2032601 |
SR1078 |
SR1078 is an agonist of retinoic acid receptor-related orphan receptor α/γ (RORα
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R2032602 |
JNJ1661010 |
JNJ-1661010 (Takeda-25) a potent and selective fatty acid amide hydrolase (FAAH)
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R2032603 |
SAR405838(MI-773) |
SAR405838 is a highly potent and selective MDM2 inhibitor, binds to MDM2 with Ki
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R2032604 |
4E1RCat |
4E1RCat is an inhibitor of cap-dependent translation, and inhibits eIF4E:eIF4GI
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R2032605 |
Salirasib |
Salirasib is a Ras inhibitor that inhibits specifically both oncogenically activ
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R2032606 |
WEHI539 |
WEHI-539 is a selective inhibitor of Bcl-XL with an IC50 of 1.1 nM.
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R2032607 |
GSK1324726A(I-BET726) |
GSK1324726A is a novel, potent, and selective inhibitor of BET proteins with hig
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R2032608 |
GSK-LSD1 2HCl |
GSK-LSD1 2HCl is an irreversible, and selective LSD1 inhibitor with IC50 of 16 n
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R2032609 |
Afuresertib(GSK2110183) |
GSK2110183 analog 1 is the structural analogue of GSK2110183.
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R2032610 |
ORG27569 |
Org 27569 is a potent CB1 receptor allosteric modulator, which increases agonist
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R2032611 |
NVP-231 |
NVP-231 is a potent, specific, and reversible CerK inhibitor(IC50=12±2 nM) that
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R2032612 |
b-AP15;NSC 687852) |
b-AP15 is a specific inhibitor of the deubiquitinating enzymes UCHL5 and Usp14.
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R2032613 |
AZ5104 |
AZ-5104 is an active, demethylated metabolite of AZD 9291.AZ-5104 is an EGFR inh
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R2032614 |
Cathepsin S inhibitor |
LY 3000328 is a potent and selective Cathepsin S (Cat S) inhibitor with IC50s of
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R2032615 |
GSK1014802(CNV1014802) |
Raxatrigine (GSK-1014802) is a novel small molecule state-dependent sodium chann
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