R2032617 |
GSK650394 |
GSK 650394 is a novel SGK inhibitor with IC50 of 62 nM and 1
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R2032618 |
INCB032304 |
INCB032304 is a pharmaceutical intermediate.
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R2032619 |
KRCA-0008 |
KRCA-0008 is a potent and selective ALK/Ack1 inhibitor with IC50 of 12 nM/4 nM f
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R2032620 |
LY2484595 |
Evacetrapib is a potent and selective of CETP inhibitor, which inhibits human re
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R2032621 |
RGB-286638 |
RGB-286638 is a CDK inhibitor that inhibits the kinase activity of cyclin T1-CDK
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R2032622 |
TG003 |
TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50
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R2032623 |
Thiamet G |
Thiamet G is a potent and selective inhibitor of O-GlcNAcase (OGA), which acts t
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R2032624 |
UNC0642 |
UNC0642 is a potent and selective G9a/GLP inhibitor, with an IC50 of less than 2
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R2032625 |
z-devd-fmk |
Z-DEVD-FMK is a specific and irreversible caspase-3 inhibitor with IC50 of 18 μM
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R2032626 |
BMS663068;Fostemsavir(BMS-663068) |
Fostemsavir (BMS-663068) is the phosphonooxymethyl prodrug of BMS-626529.Fostems
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R2032627 |
BX517(PDK1 inhibitor2) |
BX517 is a potent and selective inhibitor of PDK1 with IC50 of 6 nM.
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R2032628 |
Darapladib(SB-480848) |
Darapladib is a potent inhibitor of lipoprotein-associated phospholipase A2 (Lp-
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R2032629 |
GDC-0349 |
GDC-0349 is a potent and selective ATP-competitive mTOR inhibitor with a Ki of 3
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R2032630 |
GSK-J4 |
GSK-J4 is a potent dual inhibitor of H3K27me3/me2-demethylases JMJD3/KDM6B and U
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R2032631 |
GSK2838232 |
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R2032632 |
KN-92 hydrochloride |
KN-92 hydrochloride is an inactive derivative of KN-93.KN-93 is a selective inhi
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R2032633 |
KNK437 |
KNK437 is a HSP inhibitor, and inhibits the induction of HSP105, HSP70, and HSP4
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R2032634 |
Cligosiban(PF-3274167) |
Cligosiban (PF-3274167), a high oral bioavailability and good brain-penetrant no
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R2032635 |
SANT-1 |
SANT-1 is a potent Smo antagonist, inhibits Hedgehog signaling, with IC50s of 20
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R2032636 |
SB239063 |
SB 239063 is a potent, selective and orally active p38 MAPK inhibitor, exhibits
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R2032637 |
AEE788(NVP-AEE788) |
AEE788 is an inhibitor of the EGFR and ErbB2 with IC50 values of 2 and 6 nM, res
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R2032638 |
DDR1-IN-1 |
DDR1-IN-1 is a potent and selective DDR1 receptor tyrosine kinase inhibitor with
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R2032639 |
Decernotinib(VX-509) |
Decernotinib is a potent, orally active JAK3 inhibitor, with Kis of 2.5, 11, 13
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R2032640 |
EGF816;Nazartinib |
Nazartinib (EGF816) is a novel, covalent mutant-selective EGFR inhibitor, with K
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R2032641 |
GSK5959 |
GSK-5959 is a potent, selective and cell permeable BRPF1 bromodomain inhibitor w
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