R2032642 |
MK8245 |
MK-8245 is a potent, liver-targeted stearoyl-CoA desaturase (SCD) inhibitor, wit
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R2032643 |
NS6180 |
NS6180 is a novel potent and selective KCa3.1 channel inhibitor(IC50= 9 nM) prev
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R2032644 |
OF-1 |
OF-1 is a selective BRPF1B and BRPF2 bromodomain inhibitor with Kd values of 100
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R2032645 |
RQ-00203078 |
RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist
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R2032646 |
T-5224 |
T-5224 is a transcription factor c-Fos/activator protein (AP)-1 inhibitor with a
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R2032647 |
TCS5861528 |
Chembridge-5861528 is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-e
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R2032648 |
UNC0224 |
UNC0224 is a potent and selective G9a inhibitor with IC50 of 15 nM in the G9a Th
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R2032649 |
VER155008 |
VER-155008 is an inhibitor of Hsp70, with IC50s of 0.5 μM, 2.6 μM, and 2.6 μM fo
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R2032650 |
Vorapaxar;SCH530348 |
Vorapaxar (SCH 530348), an antiplatelet agent, is a selective, orally active, an
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R2032652 |
ZM447439 |
ZM-447439 is an aurora kinase inhibitor with IC50s of 110 and 130 nM for aurora
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R2032653 |
CCT244747 |
CCT244747 is a potent, orally bioavailable and highly selective CHK1 inhibitor,
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R2032654 |
AVN944 |
AVN-944(VX-944) is a selective, noncompetitive inhibitor of the enzyme directed
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R2032656 |
AZD-5597 |
AZD-5597 is potent CDK inhibitor with in vitro anti-proliferative effects agains
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R2032657 |
BET bromodomain inhibitor |
BET bromodomain inhibitor is a potent BET inhibitor extracted from patent WO/201
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R2032658 |
B-Raf inhibitor |
A Tyrosine kinase inhibitor.
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R2032659 |
BRD7552 |
BRD7552 is an inducer of transcription factor PDX1, which increases insulin expr
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R2032660 |
CAY10415;MSDC0160(Mitoglitazone) |
MSDC 0160 (Mitoglitazone) is a mitochondrial target of thiazolidinediones (mTOT)
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R2032661 |
CEP28122 |
CEP-28122 is a highly potent and selective orally active ALK inhibitor with IC50
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R2032662 |
CEP-37440 |
CEP-37440 is a novel potent and selective Dual FAK/ALK inhibitor with IC50 s of
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R2032663 |
E-64 |
E-64 (Proteinase inhibitor E 64) is a potent irreversible inhibitor against gene
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R2032664 |
EPZ011989 |
EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki <
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R2032665 |
Givinostat hydrochloride monohydrate(ITF2357) |
Givinostat hydrochloride monohydrate (ITF-2357 hydrochloride monohydrate) is a H
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R2032666 |
HA130 |
HA130 is a selective autotaxin (ATX) inhibitor with an IC50 of 28 nM.
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R2032667 |
LY3009120 |
LY3009120 is a pan RAF inhibitor which inhibits BRAFV600E, BRAFWT and CRAFWT wit
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R2032668 |
MK-5108(VX-689) |
MK-5108 is a highly potent and specific inhibitor of Aurora A kinase with an IC5
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