R2032669 |
ORY-1001 dihydrochloride(RG-6016) |
ORY-1001 (RG-6016) 2HCl is an orally active and selective lysine-specific demeth
|
R2032670 |
PCI-27483 |
PCI-27483 is a FVIIa/tissue factor inhibitor, with antitumour effects.
|
R2032671 |
PD123319 |
PD 123319 (ditrifluoroacetate) is a potent, selective AT2 angiotensin II recepto
|
R2032673 |
Pyroxamide |
Pyroxamide is a potent inhibitor of histone deacetylase 1 (HDAC1) with an ID50 o
|
R2032674 |
SB-399885 |
SB399885 is a potent, selective, brain penetrant and orally active 5-HT6 recepto
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R2032675 |
SB-590885 |
SB-590885 is a potent B-Raf inhibitor with Ki of 0.16 nM, and has 11-fold greate
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R2032676 |
Volasertib(BI6727) |
Volasertib is a highly potent Polo-like kinase 1 (PLK1) inhibitor with an IC50 o
|
R2032677 |
VX-11e |
VX-11e is a potent, selective, and orally bioavailable inhibitor of ERK with Ki
|
R2032678 |
AMG337 |
AMG-337 is a potent and highly selective small molecule ATP-competitive MET kina
|
R2032679 |
AZD3264 |
AZD3264 is a selective IkB-kinase IKK2 inhibitor.
|
R2032680 |
AZD8835 |
AZD8835 is a potent and selective inhibitor of PI3Kα and PI3Kδ with IC50s of 6.2
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R2032682 |
BPTES |
BPTES is an allosteric and selective glutaminase inhibitor with an IC50 of 0.16
|
R2032683 |
Pitolisant HCL |
Pitolisant hydrochloride is a potent and selective nonimidazole inverse agonist
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R2032684 |
Conduritol B epoxide |
Conduritol B epoxide is an irreversible covalently bound acid β-glucosidase (GCa
|
R2032685 |
DASA-58 |
DASA-58 is a potent activator of pyruvate kinase M2 (PKM2) with an AC90 of 680 n
|
R2032686 |
Firategrast(SB683699) |
Firategrast is an orally bioavailable α4β1/α4β7 integrin antagonist.
|
R2032687 |
GSK1070916 |
GSK-1070916 is a potent and selective ATP-competitive inhibitor of aurora B and
|
R2032688 |
GSK1278863;Daprodustat |
Daprodustat (GSK1278863) is an orally active hypoxia-inducible factor prolyl hyd
|
R2032689 |
JNJ-42041935 |
JNJ-42041935 is a potent, competitive and selective inhibitor of prolyl hydroxyl
|
R2032690 |
Ki20227 |
Ki20227 is an orally active and highly selective c-Fms tyrosine kinase (CSF1R) i
|
R2032691 |
KW2449 |
KW-2449 is a multi-targeted kinase inhibitor of FLT3, ABL, ABLT315I and Aurora k
|
R2032692 |
LDN-214117 |
LDN-214117 is a potent and selective ALK2 inhibitor with IC50 of 22 nM; > 100
|
R2032693 |
ML224(NCGC00242364;ANTAG3) |
ML224(NCGC00242364; ANTAG3) is a selective TSHR inverse agonist; inhibits TSH-st
|
R2032694 |
NVP-BHG712 |
NVP-BHG712 is an oral active EphB4 kinase autophosphorylation inhibitor, with IC
|
R2032695 |
NVP-BSK805 |
NVP-BSK805 (BSK 805) is an ATP-competitive JAK2 inhibitor, with IC50s of 0.48 nM
|