R2032696 |
PF-04457845 |
PF-04457845 is a highly efficacious and selective FAAH inhibitor with IC50 value
|
R2032697 |
PF-4989216 |
PF-4989216 is a potent and selective PI3Kα inhibitor with a Ki of 0.6 nM.
|
R2032698 |
Pyridone6 |
Pyridone 6 is a pan-JAK inhibitor, which potently inhibits the JAK kinase family
|
R2032699 |
R1530 |
R1530 is the multikinase inhibitor with potential antiangiogenesis and antineopl
|
R2032700 |
RO4987655(CH-4987655) |
RO4987655 is an orally active and highly selective MEK inhibitor with an IC50 of
|
R2032701 |
Selinexor(KPT-330) |
Selinexor (KPT-330), analog of KPT-185, is an orally bioavailable selective CRM1
|
R2032702 |
SU5614 |
SU5614 is a potent and selective FLT3 inhibitor.SU5614 has inhibitory activity f
|
R2032703 |
TRAM-34 |
TRAM-34 is a highly selective blocker of intermediate-conductance calcium-activa
|
R2032704 |
A-1210477 |
A-1210477 is a potent and selective inhibitor of MCL-1 with a Ki of 0.45 nM.
|
R2032705 |
TAK-063;Balipodect |
Balipodect (TAK-063) is a highly potent, selective and orally active PDE10A inhi
|
R2032706 |
UNC0646 |
UNC0646 is a potent and selective G9a inhibitor with IC50 of 6 nM.IC50 value: 6
|
R2032707 |
HO-3867 |
HO-3867 is a selective and potent STAT3 inhibitor and shows good antitumor activ
|
R2032708 |
PFI-4 |
PFI-4 is a potent and selective and cell permeable BRPF1 bromodomain inhibitor (
|
R2032709 |
TCS359 |
TCS 359, a 2-acylaminothiophene-3-carboxamide, is a potent inhibitor of FLT3 wit
|
R2032710 |
LJH685 |
LJH685 is a potent, specific and selective RSK inhibitor, inhibits RSK1, 2, and
|
R2032711 |
LJI308 |
LJI308 is a new and potent pan-RSK inhibitor, with IC50 of 6 nM, 4 nM, and 13 nM
|
R2032712 |
AS703026;Pimasertib |
Pimasertib (AS703026) is a highly selective, potent, ATP non-competitive alloste
|
R2032713 |
Solcitinib;GSK-2586184;GLPG-0778) |
Solcitinib is an orally active, competitive, potent, selective JAK1 inhibitor, w
|
R2032714 |
A-366 |
A-366 is a potent histone methyltransferase G9a inhibitor with an IC50 of 3.3 nM
|
R2032715 |
AZ6102 |
AZ6102 is a potent dual TNKS1 and TNKS2 inhibitor, with IC50s of 3 nM and 1 nM,
|
R2032716 |
BI-7273 |
BI-7273 is a selective, and cell-permeable BRD9 inhibitor, with an IC50 and a Kd
|
R2032717 |
FIIN-3 |
FIIN-3 is an irreversible inhibitor of FGFR with an IC50 of 13.1, 21, 31.4, and
|
R2032718 |
Glutaminase C-IN-1(968) |
Glutaminase C-IN-1 (Compound 968) is an allosteric inhibitor of Glutaminase C th
|
R2032719 |
GSK-2881078 |
GSK 2881078 is a selective androgen receptor modulator potentially for the treat
|
R2032720 |
I-BRD9 |
I-BRD9 is the first selective cellular chemical probe for BRD9 (pIC50=7.3).IC50
|