R2032721 |
LDC000067 |
LDC000067 is a highly specific CDK9 inhibitor with an IC50 value of 44±10 nM in
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R2032722 |
MI-136 |
MI-136 inhibits DHT-induced expression of androgen receptor (AR) target genes.Ta
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R2032723 |
Naloxegol oxalate;NKTR-118 oxalate;AZ-13337019 oxalate) |
Naloxegol oxalate (NKTR-118 oxalate; AZ-13337019 oxalate) is an opioid-receptor
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R2032724 |
ns11021 |
NS 11021 is a potent and specific Ca2-activated big-conductance K+ Channels (KCa
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R2032725 |
NSC348884 |
NSC348884 is a nucleophosmin inhibitor disrupts oligomer formation and induces a
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R2032726 |
Obatoclax Mesylate(GX15-070 Mesylate) |
Obatoclax Mesylate (GX15-070 Mesylate) is an inhibitor of the BCL-2 family prote
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R2032727 |
PF-04929113(SNX-5422) |
SNX-5422 (PF-04929113), a prodrug of SNX-2112, is an orally active Hsp90 inhibit
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R2032728 |
PH797804 |
PH-797804 is a ATP-competitive, selective p38α/p38β inhibitor (IC50=26 nM and Ki
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R2032729 |
PIK-293 |
PIK-293 is a PI3K inhibitor, mostly for PI3Kδ with IC50 of 0.24 μM, 500-, 100- a
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R2032730 |
RBC8 |
RBC8 is a novel small molecule inhibitor of Ral GTPase; has IC50 of 3.5 μM in H2
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R2032731 |
RO31-8220 mesylate |
Ro 31-8220 mesylate is a potent PKC inhibitor, with IC50s of 5, 24, 14, 27, 24 a
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R2032732 |
SGI-7079 |
SGI-7079 is an Axl inhibitor, significantly inhibits the proliferation of SUM149
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R2032733 |
UNC1079 |
UNC1079 is the piperidine analog of UNC1021, as a structurally similar but signi
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R2032734 |
Uprosertib;GSK2141795 |
Uprosertib (GSK2141795) is a potent and selective pan-Akt inhibitor with IC50 va
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R2032735 |
vacquinol-1 |
Vacquinol-1 is an MKK4 activator, which rapidly and selectively induces glioma c
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R2032736 |
10058-F4 |
10058-F4 is a c-Myc inhibitor that prevents c-Myc-Max dimerization and transacti
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R2032737 |
AAL-993 |
AAL-993 is a highly potent inhibitor of VEGFR-1 (IC50 =130nM), VEGFR-2 (IC50=23n
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R2032739 |
AZD8330 |
AZD8330 (ARRY-424704) is a potent, uncompetitive MEK1/MEK2 inhibitor, with an IC
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R2032740 |
BAY80-6946(Copanlisib) |
Copanlisib (BAY 80-6946) is a potent, selective and ATP-competitive pan-class I
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R2032741 |
ClozapineN-Oxide |
Clozapine (N-oxide) is a pharmacologically inert metabolite of Clozapine, an ant
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R2032742 |
CP21R7 |
CP21R7 is potent GSK-3β inhibitor, with an IC50 of 1.8 nM; CP21R7 also shows inh
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R2032743 |
Evatanepag;CP-533536 |
Evatanepag (CP-533536) is an EP2 receptor selective prostaglandin E2 (PGE2) agon
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R2032744 |
CP-724714 |
CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >
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R2032745 |
DB07268 |
DB07268 is a potent and selective JNK1 inhibitor with an IC50 value of 9 nM.
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R2032747 |
GSK-J1 |
GSK-J1 is a potent inhibitor of H3K27me3/me2-demethylases JMJD3/KDM6B and UTX/KD
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