R2033024 |
Takeda-6d |
Takeda-6d has potent inhibitory activity in both B-RAF with an IC50 of 7.0 nM an
|
R2033025 |
AZ3451 |
AZ3451 is a potent protease-activated receptor-2 (PAR2) antagonist with IC50 of
|
R2033026 |
Acumapimod |
Acumapimod (BCT197) is an orally active p38 MAP kinase inhibitor, with an IC50 o
|
R2033027 |
AZD7986 |
AZD7986 is a Dipeptidyl peptidase 1 (DPP1) inhibitor with pIC50s of 6.85, 7.6, 7
|
R2033028 |
VU0155069 |
VU0155069 (CAY10593), compound 69, is a selective phospholipase D1 (PLD1) inhibi
|
R2033029 |
CC671 |
CC-671 is a dual TTK protein kinase/CDC2-like kinase (CLK2) inhibitor with IC50s
|
R2033030 |
CCG215022 |
CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of
|
R2033031 |
HLCL-61 HCL |
HLCL-61 hydrochloride is a first-in-class inhibitor of protein arginine methyltr
|
R2033032 |
LMPTP inhibitor1 |
LMPTP INHIBITOR 1 is a selective inhibitor of low molecular weight protein tyros
|
R2033033 |
LY3177833 |
LY3177833 is a CDC7 and pMCM2 inhibitor with IC50 values of 3.3 nM and 290 nM, r
|
R2033034 |
NAV2729 |
NAV-2729 is a dual Arf1/Arf6 activation inhibitor.
|
R2033035 |
Porcupine-IN-1 |
Porcn-IN-1 is potent porcupine inhibitor with an IC50 of 0.5±0.2 nM.
|
R2033036 |
SB242235 |
SB-242235 is a potent and selective p38 MAP kinase inhibitor, with an IC50 of 1.
|
R2033037 |
SR9009 |
SR9009 is a REV-ERBα/β agonist with IC50s of 670 nM and 800 nM for REV-ERBα and
|
R2033038 |
Voruciclib |
Voruciclib is an orally active and selective CDK inhibitor with Ki values of 0.6
|
R2033039 |
WAY316606 |
WAY 316606 is an inhibitor of the secreted protein sFRP-1, an endogenous antagon
|
R2033040 |
XAV939 |
XAV-939 is a Wnt/β-catenin pathway inhibitor.XAV-939 stabilizes axin by inhibiti
|
R2033041 |
CID16020046 |
CID 16020046 is a potent and selective GPR55(LPI receptor) antagonist; inhibitsG
|
R2033042 |
MF63 |
MF63 is a selective mPGES-1 inhibitor with an IC50 of 0.9 nM and 1.3 nM for pig
|
R2033043 |
ML240 |
ML240 is a potent p97 inhibitor, inhibiting p97 ATPase with IC50 value of 100 nM
|
R2033044 |
AG879 |
Tyrphostin AG 879 (AG 879) is a tyrosine kinase inhibitor that inhibits TrKA pho
|
R2033045 |
BAM15 |
BAM 15 is a novel mitochondrial protonophore uncoupler.
|
R2033046 |
B-Raf inhibitor 1 dihydrochloride |
B-Raf inhibitor 1 dihydrochloride is a potent Raf kinase inhibitor with Kis of 1
|
R2033047 |
CP671305 |
CP671305 is a potent, orally active, selective inhibitor of phosphodiesterase-4-
|
R2033048 |
Flavopiridol |
Flavopiridol (Alvocidib) is a broad spectrum and competitive inhibitor of CDKs,
|