R2101132 |
RG7834 |
RG7834 (RO 7020322) is a highly selective and orally bioavailable HBV inhibitor,
|
R2101133 |
OSMI-1 |
OSMI-1 is an inhibitor of O-GlcNAc transferase (OGT).
|
R2101134 |
SEMBL |
SEMBL is a potent NF-κB inhibitor that inhibits DNA binding of NF-κB component p
|
R2101135 |
Bleomycin sulfate |
Bleomycin Sulfate, a glycopeptide antibiotic, is an anticancer agent for squamou
|
R2101136 |
Bleomycin hydrochloride |
Bleomycin hydrochloride is an antitumor antibiotic which induces apoptosis.
|
R2101137 |
Orelabrutinib |
Orelabrutinib is an orally active and irreversible inhibitor of Bruton's tyrosin
|
R2101138 |
NRC-2694 |
NRC-2694 is an antagonist of the epidermal growth factor receptor (EGFR). It has
|
R2101139 |
GSK366 |
GSK 366 is a potent kynurenine-3-monooxygenase (KMO) inhibitor (IC50s: 0.7 nM an
|
R2101140 |
AMG 232 |
AMG 232 is a potent, selective and orally available inhibitor of p53-MDM2 intera
|
R2101141 |
Indirubin |
Indirubin is a potent cyclin-dependent kinases and GSK-3β inhibitor with IC50 of
|
R2101143 |
RepSox |
RepSox is a potent and selective of the TGFβR-1/ALK5 inhibitor.
|
R2101144 |
Voxtalisib (XL765, SAR245409) |
Voxtalisib (SAR245409, XL765) is a dual inhibitor of mTOR/PI3K, mostly for p110γ
|
R2101145 |
Aliskiren |
Aliskiren is the first in a class of drugs called direct renin inhibitors.
|
R2101146 |
SAR-020106 |
SAR-020106 is an ATP-competitive, potent, and selective CHK1 inhibitor with an I
|
R2101147 |
A-893 |
A-893 is a cell-active inhibitor of Methyltransferase SMYD2, with an IC50 of 2.8
|
R2101148 |
Mirogabalin besylate |
Mirogabalin besylate is a selective and orally available ligand for the α2δ subu
|
R2101149 |
Px-104 |
(-)-PX20606 trans isomer is an agonist of FXR (EC50s: 18 and 29 nM for FXR in FR
|
R2101150 |
RUC-4 |
RUC-4 (RUC4;RUC 4) is a potent, selective, non-RGD-mimetic αIIbβ3 integrin recep
|
R2101151 |
GDC-0077 |
GDC-0077 (RG6114) is a potent, orally available, and selective inhibitor of PI3K
|
R2101152 |
CYC065;CDK259 |
CYC065 is an orally available, second-generation ATP-competitive inhibitor of CD
|
R2101153 |
LX-2761 |
LX2761 is a chemically stable and effective inhibitor against sodium-dependent g
|
R2101154 |
Baloxavir |
Baloxavir is a first-in-class cap-dependent endonuclease inhibitor of the influe
|
R2101155 |
ARS-1323 |
ARS-1323 (the racemate of ARS-1620) is a mutant K-ras G12C inhibitor extracted f
|
R2101156 |
CDDO-2-P-Im |
CDDO-3P-Im, an analog of CDDO-Imidazolide, has a chemopreventive effect. It can
|
R2101157 |
R-268712 |
R-268712 is an effective and selective inhibitor of ALK5 IC50: 2.5 nM).
|