R2101158 |
BAZ2-ICR |
BAZ2-ICR is an epigenetic chemical probe and it also is a potent, selective, cel
|
R2101159 |
QC6352 |
QC6352 is a selective and effective KDM4C inhibitor (IC50: 35 nM).
|
R2101160 |
T-26c |
T-26c is highly potent and selective matrix metalloproteinase-13 (MMP-13) inhibi
|
R2101161 |
CDDO-2-P-Im |
CDDO-2P-Im, an analog of CDDO-Imidazolide, has a chemopreventive effect. It can
|
R2101162 |
TP 235 |
CDDO-Im is an activator of Nrf2 and PPAR (Kis: 232/344 nM for PPARα/PPARγ).
|
R2101163 |
BAY 299 |
BAY-299 is a very potent inhibitor. For BRPF2 bromodomains (BD), TAF1 BD2, TAF1L
|
R2101164 |
BMS-955176;GSK3532795 |
GSK3532795 is a potent, orally active, second-generation HIV-1 maturation inhib
|
R2101165 |
Quarfloxin |
Quarfloxin is a fluoroquinolone derivative with antineoplastic activity with IC5
|
R2101166 |
BI-3802 |
BI-3802 is a highly effective BCL6 depressant, which can inhibit the BTB domain
|
R2101167 |
GSK-484 |
GSK484 is a potent PAD-4 inhibitor (Protein-arginine deiminase type-4). GSK484 p
|
R2101168 |
BAY-850 |
BAY-850 is a potent and isoform selective ATPase family AAA domain-containing pr
|
R2101169 |
SB-204990 |
SB 204990 is an effective and specific ATP citrate lyase enzyme inhibitor.
|
R2101170 |
Quarfloxin |
Quarfloxin (CX 3543) 是一种具有抗肿瘤活性的氟喹诺酮类衍生物,其靶向抑制RNA pol I的活性,在神经母细胞瘤中的IC50 值在纳摩尔级别
|
R2101171 |
CDDO-dhTFEA (RTA dh404) |
CDDO-dhTFEA (RTA dh404), a synthetic oleanane triterpenoid compound, potently ac
|
R2101172 |
GLPG0974 |
GLPG0974 is an antagonist of free fatty acid receptor-2 (IC50: 9 nM).
|
R2101173 |
Disitertide |
Disitertide (P144) is an inhibitor of TGF-β1.
|
R2101174 |
Alantolactone |
Alantolactone(Alant camphor), a sesquiterpene lactone, has potential activity ag
|
R2101175 |
Glesatinib |
Glesatinib is an orally active and potent dual inhibitor of MET/SMO. Glesatinib
|
R2101176 |
Halofuginone |
Halofuginone,the competitive inhibitor of prolyl-tRNA synthetase(Ki=18.3 nM),cou
|
R2101177 |
UK-383367 |
UK-383367 (UK 383367) is a potent and selective inhibitor of BMP-1 (procollagen
|
R2101178 |
TP0427736 |
TP0427736 is a potent inhibitor of ALK5 kinase activity with an IC50 of 2.72 nM
|
R2101179 |
LSKL |
LSKL, Inhibitor of Thrombospondin TSP-1(TSP-1) is activation of TGF-β .
|
R2101180 |
SMAD3;SIS3 free base |
SIS3 free base is a potent and selective Smad3 phosphorylation inhibitor. SIS3 f
|
R2101181 |
Oxymatrine |
Oxymatrine is an alkaloid isolated from Sophora flavescens, used as the antibiot
|
R2101182 |
Oroxin A |
Oroxin A has antitussive and expectorant effects.
|