R912037 |
Berzosertib (Synonyms: VE-822; VX-970) |
Berzosertib (VE-822) is an ATR inhibitor with a Ki value of less than 0.2 nM. It
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R2030001 |
MDR-1339 (DWK-1339) |
MDR-1339 (DWK-1339) is an orally active and blood-brain-barrier-permeable Aβ-agg
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R2030002 |
LY2795050 |
LY2795050 is a novel selective κ-opioid Receptor (KOR) antagonist (IC50=0.72 nM)
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R2030003 |
NI-57 |
NI-57 is an inhibitor of bromodomain and plant homeodomain finger-containing (BR
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R2030004 |
Gemcabene(PD-72953) |
Gemcabene (PD-72953), a first-in-class lipid-lowering agent, lowers low-density
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R2030005 |
Calpeptin |
Calpeptin is a potent, cell penetrating calpain inhibitor, with an ID50 of 40 nM
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R2030006 |
TAS-115 mesylate (TAS-115 methanesulfonate) |
TAS-115 mesylate is a potent VEGFRand hepatocyte growth factor receptor (c-Met/H
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R2030007 |
LMP744 (MJ-III65; NSC706744) |
LMP744 (MJ-III65) is a DNA intercalator and Topoisomerase I (Top1) inhibitor wit
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R2030008 |
Indotecan (LMP-400; NSC-724998) |
Indotecan (LMP-400) is a potent topoisomerase 1(Top1) inhibitor with IC50 values
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R2030009 |
WM-8014 |
WM-8014 is an inhibitor of MOZ, a member of histone acetyltransferases, with an
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R2030010 |
PU-H71 |
PU-H71 is a potent Hsp90 inhibitor, with an IC50 of 51 nM in MDA-MB-468 cells.&n
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R2030011 |
SBI-0206965 |
SBI-0206965 is a potent, selective and cell permeable autophagy kinase ULK1 inhi
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R2030012 |
BIBR 1532 |
BIBR 1532 is a potent, selective and non-competitive telomerase inhibi
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R2030013 |
SGC2085 |
SGC2085 is a potent and selective coactivator associated arginine methyltransfer
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R2030014 |
2-D08 |
2-D08 is a cell permeable, mechanistically unique inhibitor of protein SUMOylati
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R2030015 |
SRT1720 |
SRT 1720 is a selective activator of human SIRT1 with an EC1.5 of 0.16 μM, and s
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R2030016 |
PH-002 |
PH-002 is an inhibitor of apolipoprotein (apo) E4 intramolecular domain interact
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R2030017 |
gsk583 |
GSK583 is a highly potent, orally active and selective inhibitor of RIP2 Kinase,
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R2030018 |
Purvalanol B (NG95) |
Purvalanol B(NG-95) is a cyclin-dependent kinase inhibitor with IC50 values of 6
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R2030019 |
TAS-115 |
TAS-115 is a potent VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-tar
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R2030020 |
LMP744 hydrochloride (MJ-III65 hydrochloride) |
LMP744 hydrochloride (MJ-III65 hydrochloride) is a DNA intercalator and Topoisom
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R2030021 |
Eptifibatide |
Eptifibatide is a cyclic heptapeptide, acts as a competitive antagonist for the
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R2030022 |
Liraglutide |
Liraglutide is a glucagon-like peptide-1 (GLP-1) receptor agonist used clinicall
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R2030023 |
Sermaglutide |
Semaglutide, a long-acting GLP-1 analogue, is a glucagon-like peptide-1 (GLP-1)
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R2030024 |
Glatiramer acetate |
Glatiramer acetate (also known as Copolymer 1, Cop-1, or Copaxone - as marketed
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