R910419 |
AZD-5991 Racemate |
AZD-5991 Racemate is the racemate of AZD-5991. AZD-5991 Racemate is a Mcl-1 inhi
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R910421 |
AF-353 |
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R910422 |
Gefapixant (AF219; MK-7264) |
Gefapixant is an orally active P2X3 receptor (P2X3R) antagonist with IC50s of ~3
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R910423 |
lox-292;Selpercatinib |
Selpercatinib (LOXO-292) is a RET kinase inhibitor extracted from pate
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R910424 |
TUG-1375 |
TUG-1375 is an agonist of free fatty acid receptor 2 (FFA2/GPR43), with a pKi of
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R181104 |
BIX02188 |
BIX02188 is a selective inhibitor of MEK5 with IC50
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R912001 |
Valecobulin hydrochloride;CKD-516 hydrochloride |
Valecobulin (CKD516), a valine prodrug of (S516) and a vascular disrupting agent
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R912013 |
Fatostatin A |
Fatostatin (125B11) is an inhibitor of SREBP that directly binds SCAP and blocks
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R912018 |
Nelfinavir Mesylate (AG 1343 Mesylate) |
Nelfinavir Mesylate (AG 1343 Mesylate) is a potent and orally bioavailable HIV-1
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R912019 |
c-di-AMP (Cyclic diadenylate; Cyclic-di-AMP) |
c-di-AMP (Cyclic diadenylate) is a STING agonist, which binds to the transmembra
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R912020 |
cGAMP (Synonyms: Cyclic GMP-AMP; 3',3'-cGAMP) |
cGAMP(Cyclic GMP-AMP; 3',3'-cGAMP) is an endogenous second messenger in metazoan
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R912021 |
Sultopride hydrochloride (LIN-1418 hydrochloride) |
Sultopride hydrochloride is a selective antagonist of dopamine D2 receptor. 
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R912022 |
Zamicastat (Synonyms: BIA 5-1058) |
Zamicastat (BIA 5-1058) is a dopamine β-hydroxylase (DBH) inhibitor that could c
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R912023 |
Avacopan (CCX168) |
Avacopan (CCX168) is a potent, selective and orally available complement 5a rece
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R912025 |
LR-90 |
LR-90 is an advanced glycation end product (AGE) inhibitor, inhibits inflammator
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R912026 |
PD146176 (Synonyms: NSC168807) |
PD146176 (NSC168807) is a 15-Lipoxygenase (15-LO) inhibitor, which inhibits rabb
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R912027 |
Pralsetinib (Synonyms: BLU-667) |
Pralsetinib (BLU-667) is a highly potent, selective RET inhibitor. Pralsetinib (
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R912028 |
Atorvastatin related compound E |
N/A
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R912029 |
2-HBA |
2-HBA is a potent inducer of NAD(P)H:quinone acceptor oxidoreductase 1 (NQO1) wh
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R912030 |
CCCP (Synonyms: Carbonyl cyanide 3-chlorophenylhydrazone; Carbonyl Cyanide m-Chlorophenylhydrazone) |
CCCP is an oxidative phosphorylation uncoupler. CCCP induces activation of PINK1
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R912031 |
MRTX849 |
MRTX849 is a potent, orally-available, and mutation-selective covalent inhibitor
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R912033 |
LY2880070 |
Synonyms:(R)-[5-(2-methoxy-6-methyl-pyridin-3-yl)-2H-pyrazol-3-yl]-[6-(piperidin
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R912034 |
Lasmiditan (Synonyms: COL-144; LY573144) |
Lasmiditan (COL-144) is a high-affinity, highly selective 5-HT1F receptor agonis
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R912035 |
Lasmiditan succinate(Synonyms: COL-144 succinate; LY573144 succinate) |
Lasmiditan (COL-144) is a high-affinity, highly selective 5-HT1F receptor agonis
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R912036 |
Berzosertib hydrochloride (Synonyms: VE-822 hydrochloride; VX-970 hydrochloride) |
Berzosertib (VE-822) is an ATR inhibitor with a Ki value of less than 0.2 nM. It
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