R2030056 |
Alogliptin (SYR-322 free base) |
Alogliptin (SYR-322 free base) is a potent, selective inhibitor of DPP-4 with IC
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R2030057 |
Aceclofenac |
Aceclofenac is a non-steroidal anti-inflammatory drug (NSAID) analog of Diclofen
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R2030058 |
ASP3026 |
ASP3026 is a novel and selective inhibitor for ALK (anaplastic lymphoma kinase)
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R2030059 |
Mutant EGFR inhibitor |
Mutant EGFR inhibitor is a potent and selective mutant EGFR inhibitor extracted
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R2030060 |
Rociletinib hydrobromide(CO-1686 hydrobromide;AVL-301 hydrobromide;CNX-419 hydrobromide) |
Rociletinib hydrobromide (CO-1686 hydrobromide) is an orally delivered kinase in
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R2030061 |
JAK3-IN-1 |
JAK3-IN-1 (Compound 9) is a potent, selective and orally active JAK3 inhibitor w
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R2030062 |
Amcasertib (BBI503) |
Amcasertib is an orally administered investigational agent designed to inhibit c
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R2030063 |
BACE1-IN-2 |
BACE1-IN-2 is a 1,4-Oxazine β-Secretase 1 (BACE1) inhibitor with an IC50 of 22 n
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R2030064 |
JNJ-678 (JNJ-53718678) |
JNJ-678 (JNJ-53718678) is a novel fusion protein inhibitor in clinical trials fo
|
R2030065 |
IDO-IN-8 (NLG-1487) |
IDO-IN-8 (NLG-1487) is an indoleamine 2,3-dioxygenase (IDO) inhibitor extracted
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R2030066 |
GSK2798745 |
GSK2798745 is a first-in-class, highly potent, selective, orally active transien
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R2030067 |
Zoliflodacin (ETX0914; AZD0914) |
Zoliflodacin (ETX0914;AZD0914) is a novel spiropyrimidinetrione bacterial DNA gy
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R2030068 |
Enasidenib mesylate (AG-221 mesylate) |
Enasidenib mesylate is a first-in-class, oral, potent, reversible, selective inh
|
R2030069 |
CM-4620 |
CM-4620 is a calcium-release activated calcium-channel (CRAC channel) inhibitor,
|
R2030070 |
PF-06650833 |
PF06650833 is a potent, selective and orally active inhibitor of interleukin-1 r
|
R2030071 |
PF-06840003 (EOS200271) |
PF-06840003 is a highly selective orally bioavailable IDO-1 inhibitor with
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R2030072 |
Agerafenib (CEP-32496; RXDX-105) |
Agerafenib (CEP-32496; RXDX-105) is a highly potent and orally efficacious inhib
|
R2030073 |
Capivasertib (AZD5363) |
Capivasertib (AZD5363) is a potent pan-AKT kinase inhibitor with IC50 of 3, 7 an
|
R2030074 |
CDM-NAG |
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R2030075 |
Miridesap (CPHPC; Ro63-8695; GSK2315698) |
Miridesap is a ligand for serum amyloid P component (SAP) and intends to inhibit
|
R2030076 |
Afuresertib (GSK2110183) |
Afuresertib (GSK2110183) is an orally bioavailable, selective, ATP-competitive a
|
R2030077 |
GSK2879552 |
GSK2879552 is an orally available, irreversible inhibitor of lysine specific dem
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R2030078 |
IB-MECA acetonide |
IB-MECA acetonide is an agonist of the adenosine A3 receptor with EC50 valu
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R2030079 |
IDO-IN-7;Navoximod (GDC-0919; NLG-919) |
Navoximod (GDC-0919; NLG-919) is a potent IDO (indoleamine-(2,3)-dioxygenase) p
|
R2030081 |
LUF6000 |
LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR). IC50
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