R2030113 |
Imidazole ketone erastin (IKE) |
Imidazole ketone erastin (IKE) is a potent, selective, and metabolically stable
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R2030114 |
L-779450 |
L-779450 is a potent and selective B-Raf kinase inhibitor with a Kd of 2.4 nM.&n
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R2030116 |
TAK-981;TAK981 |
TAK-981 is a first in class and selective inhibitor of the SUMOylation enzymatic
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R2030117 |
AZ505 |
AZ505 is a potent and selective SMYD2 inhibitor with IC50 of 0.12 μM.
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R2030118 |
BAY-598 |
BAY-598 is selective small molecule inhibitor of SMYD2 with an IC50 of 27 nM.
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R2030119 |
CTEP (RO 4956371; mGluR5 inhibitor) |
CTEP (RO 4956371) is a novel, long-acting, orally bioavailable allosteric antago
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R2030120 |
Basimglurant (RG7090; CTEP Derivative) |
Basimglurant (RG7090) is a potent, selective and orally available mGlu5 negative
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R2030121 |
D-Luciferin |
D-luciferin is the natural substrate of luciferases that catalyze the production
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R2030124 |
LDN-192960 |
LDN-192960 is an inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kin
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R2030125 |
Motesanib Diphosphate (AMG-706) VM-2005 |
Motesanib Diphosphate (AMG 706 Diphosphate) is a potent ATP-competitive inhibito
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R2030126 |
PTC-209 |
PTC-209 is a specific BMI-1 inhibitor with an IC50 of 0.5 μM.
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R2030127 |
SMI-4a |
(Z)-SMI-4a is a poten, selective, cell-permeable and ATP-competitive Pim-1 inhib
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R2030128 |
SU-9516 |
SU9516 is a potent CDK2 inhibitor, with an IC50 of 22 nM, and also shows inhibit
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R2030129 |
TDZD-8 (GSK-3β Inhibitor I; NP 01139) |
TDZD-8 is an inhibitor of GSK-3β, with an IC50 of 2 μM; TDZD-8 shows less potent
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R2030130 |
UNC-669 |
UNC 669 is a potent antagonist of L3MBTL1(IC50=4.2 uM) and L3MBTL3(IC50=3.1 uM).
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R2030131 |
WZ-811 |
WZ811 is an orally active, highly potent competitive antagonist of CXCR4. WZ811
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R2030132 |
Rilpivirine (R278474; TMC278; DB08864) |
Rilpivirine (R278474; TMC278) is a type of anti-HIV medicine called a non-nucleo
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R2030133 |
IM-12 |
IM-12 is an inhibitor of GSK-3β, with an IC50 of 53 nM, and also enhances Wnt si
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R2030134 |
Losmapimod (GSK-AHAB; GW856553X; SB856553) |
Losmapimod is a selective, potent, and orally active p38 MAPK inhibitor with pKi
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R2030135 |
BH3I-1 (BHI1; BH 3I1) |
BH3I-1 is a Bcl-2 family antagonist, which inhibits the binding of the Bak BH3 p
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R2030136 |
IQ-1S free acid |
IQ-1S free acid is a prospective inhibitor of NF-κB/activating protein 1 (AP-1)
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R2030137 |
IQ 1 |
IQ 1 has many functions such as decreasing Wnt-stimulated phosphorylation, maint
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R2030138 |
A804598 |
A-804598 is a CNS penetrant, competitive and selective P2X7 receptor antagonist
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R2030139 |
Pifithrin-α hydrobromide (Pifithrin hydrobromide; PFTα hydrobromide) |
Pifithrin-α hydrobromide is a p53 inhibitor which blocks its transcriptional act
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R2030140 |
HMN-176 |
HMN-176 is a stilbene derivative which inhibits mitosis, interfering with p
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