R2032329 |
A66 |
A66 is a highly specific and selective p110α inhibitor with an IC50 of 32 nM.
|
R2032330 |
A-674563 |
A-674563 is a potent and selective Akt1 inhibitor with a Ki of 11 nM.
|
R2032331 |
A-740003 |
A-740003 is a potent, selective and competitive P2X7 receptor antagonist with IC
|
R2032332 |
A-966492 |
A-966492 is a novel and potent inhibitor of PARP1 and PARP2 with Ki of 1 nM and
|
R2032333 |
ABT-346 |
ATB-346 is a novel hydrogen sulphide-releasing derivative of naproxen with marke
|
R2032334 |
ABT-751(E7010) |
ABT-751(E 7010) is a novel bioavailable tubulin-binding and antimitotic sulfonam
|
R2032335 |
AdipoRon |
AdipoRon is an orally active adiponectin receptor (AdipoR) agonist, binding to A
|
R2032336 |
ADL5859 |
ADL5859 is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against op
|
R2032337 |
AG1024(Tyrphostin AG 1024) |
AG1024 (Tyrphostin AG 1024) is a reversible, competitive and selective insulin-l
|
R2032338 |
AM251 |
AM251 is a selective cannabinoid 1 (CB1) receptor antagonist with an IC50 of 8 n
|
R2032339 |
AM-281;AM281 |
Potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values
|
R2032340 |
AMG837 |
AMG 837 is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic pr
|
R2032341 |
AMG900 |
AMG 900 is a potent and highly selective pan-Aurora kinases inhibitor with IC50
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R2032342 |
AT13148 |
AT13148 is an orally active and ATP-competitive, multi-AGC kinase inhibitor with
|
R2032343 |
AT-7867 |
AT7867 is a potent ATP-competitive inhibitor of Akt1/Akt2/Akt3 and p70S6K/PKA wi
|
R2032344 |
Avelestat(AZD9668) |
Alvelestat (AZD9668) is an orally bioavailable, affinity and selective inhibitor
|
R2032345 |
AVP-AEW541;AEW541 |
NVP-AEW541 is a potent inhibitor of IGF-1R with IC50 of 0.15 μM, also inhibits I
|
R2032346 |
AZ191 |
AZ191 is a potent inhibitor that selectively inhibits DYRK1B with IC50 of 17 nM.
|
R2032347 |
AZ20 |
AZ20 is a potent and selective inhibitor of ATR with an IC50 of 5 nM, and has 8-
|
R2032348 |
AZ3146 |
AZ3146 is a reasonably potent and selective Mps1 inhibitor with IC50 of 35 nM fo
|
R2032349 |
AZ960 |
AZ960 is a potent and specific inhibitor of the JAK2 kinase with a Ki of 0.45 nM
|
R2032350 |
Barasertib-HQPA;AZD2811;INH-34;AZD1152-HQPA |
Barasertib-HQPA (AZD2811) is a highly selective Aurora B inhibitor with an IC50
|
R2032351 |
AZD1208 |
AZD1208 is a novel, orally bioavailable, highly selective PIM kinases inhibitor.
|
R2032352 |
AZD1283 |
AZD1283 is a potent antagonist of the P2Y12 receptor with EC50 of 3.0 ug/kg/min,
|
R2032353 |
Vistusertib (AZD2014) |
Vistusertib (AZD2014) is an ATP competitive mTOR inhibitor with an IC50 of 2.81
|