R2032354 |
AZD2932 |
AZD2932 is a potent and multi-targeted kinase inhibitor VEGFR2, PDGFβ, Flt-3 and
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R2032355 |
AZD3514 |
AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM a
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R2032356 |
AZD6482;AZD 6482 (KIN-193) |
AZD 6482 (KIN-193) is a potent and selective p110β inhibitor with an IC50 of 0.6
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R2032357 |
AZD7545 |
AZD7545 is a potent, competitive, selective PDHK2 (pyruvate dehydrogenase kinase
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R2032358 |
BAM7 |
BAM7 is a direct and selective activator of proapoptotic BAX with an IC50 of 3.3
|
R2032359 |
BAY11-7085;BAY 11-7083 |
BAY 11-7085 is an inhibitor of NF-κB activation and phosphorylation of IκBα; it
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R2032360 |
BAY87-2243 |
BAY 87-2243 is a highly potent and selective hypoxia-inducible factor-1 (HIF-1)
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R2032361 |
Dactolisib;BEZ235;NVP-BEZ235 |
Dactolisib (BEZ235) is a dual pan-class I PI3K and mTOR kinase inhibitor with IC
|
R2032362 |
BIBX1382;Falnidamol(BIBX 1382) |
Falnidamol (BIBX 1382) is an orally active, selective EGFR tyrosine kinase inhib
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R2032363 |
GSK 3 Inhibitor IX;MLS2052 |
GSK 3 Inhibitor IX (6-Bromoindirubin-3'-oxime; BIO) is a potent, selective, reve
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R2032364 |
BIX02189 |
BIX02189 is a selective inhibitor of MEK5 with IC50 of 1.5 nM, also inhibits ERK
|
R2032365 |
BMS265246 |
BMS-265246 is a potent and selective CDK1/2 inhibitor for CDK1/cyclin B and CDK2
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R2032366 |
BMS345541 |
BMS-345541 is a selective inhibitor of the catalytic subunits of IKK (IKK-2 IC50
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R2032367 |
BMS754807 |
BMS-754807 is a potent and reversible inhibitor of IGF-1R/IR with IC50 of 1.8 an
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R2032368 |
AZD1480 |
AZD-1480 is an ATP-competitive inhibitor of JAK1 and JAK2 with IC50s of 1.3 and
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R2032369 |
BMS777607;BMS-777607;BMS 817378 |
BMS 777607 is a Met-related inhibitor for c-Met, Axl, Ron and Tyro3 with IC50s o
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R2032370 |
BMY7378 Dihydrochloride |
BMY 7378 is a multi-targeted inhibitor of α2C-adrenoceptor and α1D-adrenoceptor
|
R2032371 |
BRD4770 |
BRD4770 is a novel G9a(EHMT2) inhibitor with EC50 of 5 uM (trimethylated H3K9 in
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R2032372 |
BTB06584 |
BTB06584 is an IF1-dependent selective inhibitor of the mitochondrial F1Fo-ATPas
|
R2032373 |
BX-795 |
BX795 is a potent and selective inhibitor of PDK1, with an IC50 of 6 nM.BX795 is
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R2032374 |
BX-912 |
BX-912 is a direct, selective, and ATP-competitive PDK1 inhibitor (IC50=26 nM).B
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R2032375 |
Telaglenastat(CB-839) |
Telaglenastat (CB-839) is a first-in-class, reversible and orally bioavailable g
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R2032376 |
CCT007093 |
CCT007093 is an effective PPM1D inhibitor that selectively reduces viability of
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R2032377 |
Delanzomib(CEP-18770) |
Delanzomib(CEP-18770) is a novel orally-active inhibitor of the chymotrypsin-lik
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R2032378 |
CH5132799 |
CH5132799 is a selective class I PI3K inhibitor.CH5132799 inhibits class I PI3Ks
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