R2032604 |
4E1RCat |
4E1RCat is an inhibitor of cap-dependent translation, and inhibits eIF4E:eIF4GI
|
R2032605 |
Salirasib |
Salirasib is a Ras inhibitor that inhibits specifically both oncogenically activ
|
R2032606 |
WEHI539 |
WEHI-539 is a selective inhibitor of Bcl-XL with an IC50 of 1.1 nM.
|
R2032607 |
GSK1324726A(I-BET726) |
GSK1324726A is a novel, potent, and selective inhibitor of BET proteins with hig
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R2032608 |
GSK-LSD1 2HCl |
GSK-LSD1 2HCl is an irreversible, and selective LSD1 inhibitor with IC50 of 16 n
|
R2032609 |
Afuresertib(GSK2110183) |
GSK2110183 analog 1 is the structural analogue of GSK2110183.
|
R2032610 |
ORG27569 |
Org 27569 is a potent CB1 receptor allosteric modulator, which increases agonist
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R2032611 |
NVP-231 |
NVP-231 is a potent, specific, and reversible CerK inhibitor(IC50=12±2 nM) that
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R2032612 |
b-AP15;NSC 687852) |
b-AP15 is a specific inhibitor of the deubiquitinating enzymes UCHL5 and Usp14.
|
R2032613 |
AZ5104 |
AZ-5104 is an active, demethylated metabolite of AZD 9291.AZ-5104 is an EGFR inh
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R2032614 |
Cathepsin S inhibitor |
LY 3000328 is a potent and selective Cathepsin S (Cat S) inhibitor with IC50s of
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R2032615 |
GSK1014802(CNV1014802) |
Raxatrigine (GSK-1014802) is a novel small molecule state-dependent sodium chann
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R2032616 |
GSK503 |
GSK503 is a potent and specific inhibitor of EZH2 methyltransferase with Ki
|
R2032617 |
GSK650394 |
GSK 650394 is a novel SGK inhibitor with IC50 of 62 nM and 1
|
R2032618 |
INCB032304 |
INCB032304 is a pharmaceutical intermediate.
|
R2032619 |
KRCA-0008 |
KRCA-0008 is a potent and selective ALK/Ack1 inhibitor with IC50 of 12 nM/4 nM f
|
R2032620 |
LY2484595 |
Evacetrapib is a potent and selective of CETP inhibitor, which inhibits human re
|
R2032621 |
RGB-286638 |
RGB-286638 is a CDK inhibitor that inhibits the kinase activity of cyclin T1-CDK
|
R2032622 |
TG003 |
TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50
|
R2032623 |
Thiamet G |
Thiamet G is a potent and selective inhibitor of O-GlcNAcase (OGA), which acts t
|
R2032624 |
UNC0642 |
UNC0642 is a potent and selective G9a/GLP inhibitor, with an IC50 of less than 2
|
R2032625 |
z-devd-fmk |
Z-DEVD-FMK is a specific and irreversible caspase-3 inhibitor with IC50 of 18 μM
|
R2032626 |
BMS663068;Fostemsavir(BMS-663068) |
Fostemsavir (BMS-663068) is the phosphonooxymethyl prodrug of BMS-626529.Fostems
|
R2032627 |
BX517(PDK1 inhibitor2) |
BX517 is a potent and selective inhibitor of PDK1 with IC50 of 6 nM.
|
R2032628 |
Darapladib(SB-480848) |
Darapladib is a potent inhibitor of lipoprotein-associated phospholipase A2 (Lp-
|