R2032654 |
AVN944 |
AVN-944(VX-944) is a selective, noncompetitive inhibitor of the enzyme directed
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R2032655 |
AZD2461 |
AZD-2461 is a potent PARP inhibitor, with IC50s of 5 nM, 2 nM and 200 nM for PAR
|
R2032656 |
AZD-5597 |
AZD-5597 is potent CDK inhibitor with in vitro anti-proliferative effects agains
|
R2032657 |
BET bromodomain inhibitor |
BET bromodomain inhibitor is a potent BET inhibitor extracted from patent WO/201
|
R2032658 |
B-Raf inhibitor |
A Tyrosine kinase inhibitor.
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R2032659 |
BRD7552 |
BRD7552 is an inducer of transcription factor PDX1, which increases insulin expr
|
R2032660 |
CAY10415;MSDC0160(Mitoglitazone) |
MSDC 0160 (Mitoglitazone) is a mitochondrial target of thiazolidinediones (mTOT)
|
R2032661 |
CEP28122 |
CEP-28122 is a highly potent and selective orally active ALK inhibitor with IC50
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R2032662 |
CEP-37440 |
CEP-37440 is a novel potent and selective Dual FAK/ALK inhibitor with IC50 s of
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R2032663 |
E-64 |
E-64 (Proteinase inhibitor E 64) is a potent irreversible inhibitor against gene
|
R2032664 |
EPZ011989 |
EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki <
|
R2032665 |
Givinostat hydrochloride monohydrate(ITF2357) |
Givinostat hydrochloride monohydrate (ITF-2357 hydrochloride monohydrate) is a H
|
R2032666 |
HA130 |
HA130 is a selective autotaxin (ATX) inhibitor with an IC50 of 28 nM.
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R2032667 |
LY3009120 |
LY3009120 is a pan RAF inhibitor which inhibits BRAFV600E, BRAFWT and CRAFWT wit
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R2032668 |
MK-5108(VX-689) |
MK-5108 is a highly potent and specific inhibitor of Aurora A kinase with an IC5
|
R2032669 |
ORY-1001 dihydrochloride(RG-6016) |
ORY-1001 (RG-6016) 2HCl is an orally active and selective lysine-specific demeth
|
R2032670 |
PCI-27483 |
PCI-27483 is a FVIIa/tissue factor inhibitor, with antitumour effects.
|
R2032671 |
PD123319 |
PD 123319 (ditrifluoroacetate) is a potent, selective AT2 angiotensin II recepto
|
R2032672 |
PHA767491 |
PHA-767491 is a dual Cdc7/Cdk9 inhibitor, with IC50s of 10 nM and 34 nM, respect
|
R2032673 |
Pyroxamide |
Pyroxamide is a potent inhibitor of histone deacetylase 1 (HDAC1) with an ID50 o
|
R2032674 |
SB-399885 |
SB399885 is a potent, selective, brain penetrant and orally active 5-HT6 recepto
|
R2032675 |
SB-590885 |
SB-590885 is a potent B-Raf inhibitor with Ki of 0.16 nM, and has 11-fold greate
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R2032676 |
Volasertib(BI6727) |
Volasertib is a highly potent Polo-like kinase 1 (PLK1) inhibitor with an IC50 o
|
R2032677 |
VX-11e |
VX-11e is a potent, selective, and orally bioavailable inhibitor of ERK with Ki
|
R2032678 |
AMG337 |
AMG-337 is a potent and highly selective small molecule ATP-competitive MET kina
|