| R2032683 |
Pitolisant HCL |
Pitolisant hydrochloride is a potent and selective nonimidazole inverse agonist
|
| R2032684 |
Conduritol B epoxide |
Conduritol B epoxide is an irreversible covalently bound acid β-glucosidase (GCa
|
| R2032685 |
DASA-58 |
DASA-58 is a potent activator of pyruvate kinase M2 (PKM2) with an AC90 of 680 n
|
| R2032686 |
Firategrast(SB683699) |
Firategrast is an orally bioavailable α4β1/α4β7 integrin antagonist.
|
| R2032687 |
GSK1070916 |
GSK-1070916 is a potent and selective ATP-competitive inhibitor of aurora B and
|
| R2032688 |
GSK1278863;Daprodustat |
Daprodustat (GSK1278863) is an orally active hypoxia-inducible factor prolyl hyd
|
| R2032689 |
JNJ-42041935 |
JNJ-42041935 is a potent, competitive and selective inhibitor of prolyl hydroxyl
|
| R2032690 |
Ki20227 |
Ki20227 is an orally active and highly selective c-Fms tyrosine kinase (CSF1R) i
|
| R2032691 |
KW2449 |
KW-2449 is a multi-targeted kinase inhibitor of FLT3, ABL, ABLT315I and Aurora k
|
| R2032692 |
LDN-214117 |
LDN-214117 is a potent and selective ALK2 inhibitor with IC50 of 22 nM; > 100
|
| R2032693 |
ML224(NCGC00242364;ANTAG3) |
ML224(NCGC00242364; ANTAG3) is a selective TSHR inverse agonist; inhibits TSH-st
|
| R2032694 |
NVP-BHG712 |
NVP-BHG712 is an oral active EphB4 kinase autophosphorylation inhibitor, with IC
|
| R2032695 |
NVP-BSK805 |
NVP-BSK805 (BSK 805) is an ATP-competitive JAK2 inhibitor, with IC50s of 0.48 nM
|
| R2032696 |
PF-04457845 |
PF-04457845 is a highly efficacious and selective FAAH inhibitor with IC50 value
|
| R2032697 |
PF-4989216 |
PF-4989216 is a potent and selective PI3Kα inhibitor with a Ki of 0.6 nM.
|
| R2032698 |
Pyridone6 |
Pyridone 6 is a pan-JAK inhibitor, which potently inhibits the JAK kinase family
|
| R2032699 |
R1530 |
R1530 is the multikinase inhibitor with potential antiangiogenesis and antineopl
|
| R2032700 |
RO4987655(CH-4987655) |
RO4987655 is an orally active and highly selective MEK inhibitor with an IC50 of
|
| R2032701 |
Selinexor(KPT-330) |
Selinexor (KPT-330), analog of KPT-185, is an orally bioavailable selective CRM1
|
| R2032702 |
SU5614 |
SU5614 is a potent and selective FLT3 inhibitor.SU5614 has inhibitory activity f
|
| R2032703 |
TRAM-34 |
TRAM-34 is a highly selective blocker of intermediate-conductance calcium-activa
|
| R2032704 |
A-1210477 |
A-1210477 is a potent and selective inhibitor of MCL-1 with a Ki of 0.45 nM.
|
| R2032705 |
TAK-063;Balipodect |
Balipodect (TAK-063) is a highly potent, selective and orally active PDE10A inhi
|
| R2032706 |
UNC0646 |
UNC0646 is a potent and selective G9a inhibitor with IC50 of 6 nM.IC50 value: 6
|
| R2032707 |
HO-3867 |
HO-3867 is a selective and potent STAT3 inhibitor and shows good antitumor activ
|