R2032704 |
A-1210477 |
A-1210477 is a potent and selective inhibitor of MCL-1 with a Ki of 0.45 nM.
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R2032705 |
TAK-063;Balipodect |
Balipodect (TAK-063) is a highly potent, selective and orally active PDE10A inhi
|
R2032706 |
UNC0646 |
UNC0646 is a potent and selective G9a inhibitor with IC50 of 6 nM.IC50 value: 6
|
R2032707 |
HO-3867 |
HO-3867 is a selective and potent STAT3 inhibitor and shows good antitumor activ
|
R2032708 |
PFI-4 |
PFI-4 is a potent and selective and cell permeable BRPF1 bromodomain inhibitor (
|
R2032709 |
TCS359 |
TCS 359, a 2-acylaminothiophene-3-carboxamide, is a potent inhibitor of FLT3 wit
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R2032710 |
LJH685 |
LJH685 is a potent, specific and selective RSK inhibitor, inhibits RSK1, 2, and
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R2032711 |
LJI308 |
LJI308 is a new and potent pan-RSK inhibitor, with IC50 of 6 nM, 4 nM, and 13 nM
|
R2032712 |
AS703026;Pimasertib |
Pimasertib (AS703026) is a highly selective, potent, ATP non-competitive alloste
|
R2032713 |
Solcitinib;GSK-2586184;GLPG-0778) |
Solcitinib is an orally active, competitive, potent, selective JAK1 inhibitor, w
|
R2032714 |
A-366 |
A-366 is a potent histone methyltransferase G9a inhibitor with an IC50 of 3.3 nM
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R2032715 |
AZ6102 |
AZ6102 is a potent dual TNKS1 and TNKS2 inhibitor, with IC50s of 3 nM and 1 nM,
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R2032716 |
BI-7273 |
BI-7273 is a selective, and cell-permeable BRD9 inhibitor, with an IC50 and a Kd
|
R2032717 |
FIIN-3 |
FIIN-3 is an irreversible inhibitor of FGFR with an IC50 of 13.1, 21, 31.4, and
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R2032718 |
Glutaminase C-IN-1(968) |
Glutaminase C-IN-1 (Compound 968) is an allosteric inhibitor of Glutaminase C th
|
R2032719 |
GSK-2881078 |
GSK 2881078 is a selective androgen receptor modulator potentially for the treat
|
R2032720 |
I-BRD9 |
I-BRD9 is the first selective cellular chemical probe for BRD9 (pIC50=7.3).IC50
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R2032721 |
LDC000067 |
LDC000067 is a highly specific CDK9 inhibitor with an IC50 value of 44±10 nM in
|
R2032722 |
MI-136 |
MI-136 inhibits DHT-induced expression of androgen receptor (AR) target genes.Ta
|
R2032723 |
Naloxegol oxalate;NKTR-118 oxalate;AZ-13337019 oxalate) |
Naloxegol oxalate (NKTR-118 oxalate; AZ-13337019 oxalate) is an opioid-receptor
|
R2032724 |
ns11021 |
NS 11021 is a potent and specific Ca2-activated big-conductance K+ Channels (KCa
|
R2032725 |
NSC348884 |
NSC348884 is a nucleophosmin inhibitor disrupts oligomer formation and induces a
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R2032726 |
Obatoclax Mesylate(GX15-070 Mesylate) |
Obatoclax Mesylate (GX15-070 Mesylate) is an inhibitor of the BCL-2 family prote
|
R2032727 |
PF-04929113(SNX-5422) |
SNX-5422 (PF-04929113), a prodrug of SNX-2112, is an orally active Hsp90 inhibit
|
R2032728 |
PH797804 |
PH-797804 is a ATP-competitive, selective p38α/p38β inhibitor (IC50=26 nM and Ki
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