R2032729 |
PIK-293 |
PIK-293 is a PI3K inhibitor, mostly for PI3Kδ with IC50 of 0.24 μM, 500-, 100- a
|
R2032730 |
RBC8 |
RBC8 is a novel small molecule inhibitor of Ral GTPase; has IC50 of 3.5 μM in H2
|
R2032731 |
RO31-8220 mesylate |
Ro 31-8220 mesylate is a potent PKC inhibitor, with IC50s of 5, 24, 14, 27, 24 a
|
R2032732 |
SGI-7079 |
SGI-7079 is an Axl inhibitor, significantly inhibits the proliferation of SUM149
|
R2032733 |
UNC1079 |
UNC1079 is the piperidine analog of UNC1021, as a structurally similar but signi
|
R2032734 |
Uprosertib;GSK2141795 |
Uprosertib (GSK2141795) is a potent and selective pan-Akt inhibitor with IC50 va
|
R2032735 |
vacquinol-1 |
Vacquinol-1 is an MKK4 activator, which rapidly and selectively induces glioma c
|
R2032736 |
10058-F4 |
10058-F4 is a c-Myc inhibitor that prevents c-Myc-Max dimerization and transacti
|
R2032737 |
AAL-993 |
AAL-993 is a highly potent inhibitor of VEGFR-1 (IC50 =130nM), VEGFR-2 (IC50=23n
|
R2032738 |
AV412 |
AV-412 free base (MP-412 free base) is an EGFR inhibitor with IC50s of 0.75, 0.5
|
R2032739 |
AZD8330 |
AZD8330 (ARRY-424704) is a potent, uncompetitive MEK1/MEK2 inhibitor, with an IC
|
R2032740 |
BAY80-6946(Copanlisib) |
Copanlisib (BAY 80-6946) is a potent, selective and ATP-competitive pan-class I
|
R2032741 |
ClozapineN-Oxide |
Clozapine (N-oxide) is a pharmacologically inert metabolite of Clozapine, an ant
|
R2032742 |
CP21R7 |
CP21R7 is potent GSK-3β inhibitor, with an IC50 of 1.8 nM; CP21R7 also shows inh
|
R2032743 |
Evatanepag;CP-533536 |
Evatanepag (CP-533536) is an EP2 receptor selective prostaglandin E2 (PGE2) agon
|
R2032744 |
CP-724714 |
CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >
|
R2032745 |
DB07268 |
DB07268 is a potent and selective JNK1 inhibitor with an IC50 value of 9 nM.
|
R2032746 |
GDC-0879 |
GDC-0879 is a potent and selective B-Raf inhibitor with an IC50 of 0.13 nM.
|
R2032747 |
GSK-J1 |
GSK-J1 is a potent inhibitor of H3K27me3/me2-demethylases JMJD3/KDM6B and UTX/KD
|
R2032748 |
MK-2461 |
MK-2461 is a novel ATP-competitive multitargeted inhibitor of activated c-Met wi
|
R2032749 |
PF8380 |
PF-8380 is a potent autotaxin inhibitor with an IC50 of 2.8 nM in isolated enzym
|
R2032750 |
PRX08066 |
PRX-08066 Maleic acid is a selective 5-HT2B receptor antagonist with IC50 of 3.4
|
R2032751 |
RO41-1049 HCL |
Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine ox
|
R2032752 |
Ro41-1049 hydrochloride |
Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine ox
|
R2032753 |
Tetrabenazine |
Tetrabenazine (Racemate) is a selective and reversible inhibitor of vesicular mo
|