R2032754 |
Vadimezan(DMXAA;ASA-404) |
Vadimezan (DMXAA; ASA-404), the tumor vascular disrupting agent (tumor-VDA), is
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R2032755 |
ms023 |
MS023 is a potent, selective, and cell-active inhibitor of human type I protein
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R2032756 |
Brincidofovir(CMX001) |
Brincidofovir (CMX001; HDP-CDV) is an orally active, lipophilic form of cidofovi
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R2032757 |
FRAX1036 |
FRAX1036 is a PAK inhibitor with Kis of 23.3 nM, 72.4 nM, and 2.4 μM for PAK1, P
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R2032758 |
Itacitinib |
Itacitinib is an orally bioavailable and selective inhibitor of JAK1, with >2
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R2032759 |
JI-101 |
JI-101 is an orally available multi-kinase inhibitor of VEGFR2,PDGFRβ and EphB4
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R2032760 |
PF2545920;Mardepodect(PF-2545920) |
Mardepodect (PF-2545920) is a potent, orally active and selective PDE10A inhibit
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R2032761 |
RPI-1 |
RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.
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R2032762 |
SNX-2112(PF-04928473) |
SNX-2112 (PF 04928473) is an orally active Hsp90 inhibitor, with a Kd of 16 nM f
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R2032763 |
AG14361 |
AG14361 is a potent PARP-1 inhibitor, with a Ki of < 5 nM, and in permeabiliz
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R2032764 |
AGK2 |
AGK2 is a selective SIRT2 inhibitor with IC50 of 3.5 μM.AGK2 can also inhibit SI
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R2032765 |
AM2394 |
AM-2394 is a structurally distinct glucokinase activator (GKA).AM-2394 activates
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R2032766 |
Bevirimat |
Bevirimat (PA-457; MPC-4326; YK FH312) is an anti-HIV drug derived from a betuli
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R2032767 |
BMS707035 |
BMS-707035 is an HIV-1 integrase (IN) inhibitor with an IC50 value of 15 nM.IC50
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R2032768 |
CDKI-73 |
CDKI-73 is a potent CDK9 inhibitor with Ki of 4 nM; shows selective toxicity to
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R2032769 |
cpi-637 |
CPI-637 is a selective and potent CBP/EP300 bromodomain inhibitor with IC50 valu
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R2032770 |
EHT1864 |
EHT 1864 is an inhibitor of Rac family small GTPases.EHT 1864 directly binds and
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R2032771 |
EPZ020411 |
EPZ020411 is a potent and selective inhibitor of PRMT6 with IC50 of 10 nM, has >
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R2032772 |
Fenebrutinib(GDC-0853) |
Fenebrutinib (GDC-0853) is a potent, selective, and noncovalent bruton's tyrosin
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R2032773 |
GGTI298 |
GGTI298 is a CAAZ peptidomimetic geranylgeranyltransferase I (GGTase I) inhibito
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R2032774 |
GSK2981278 |
GSK2981278 is a potent and selective RORγ inverse agonist.GSK2981278 inhibits ac
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R2032775 |
GSK6853 |
GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain.shows excel
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R2032776 |
ITSA-1 |
ITSA-1 is an activator of histone deacetylase (HDAC), and counteract trichostati
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R2032777 |
KN62 |
KN-62 is a selective and potent inhibitor of calmodulin-dependent protein kinase
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R2032778 |
L755507 |
L755507 is a potent, selective agonist of β3-AR with an IC50 of 35 nM.
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