R2032979 |
ABT702 dihydrochloride |
ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor (IC50=1.7 nM
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R2032980 |
BAY1436032 |
BAY-1436032 is a novel pan-mutant isocitrate dehydrogenase 1 (IDH1) inhibitor.
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R2032981 |
CH-223191 |
CH-223191 is a potent and specific antagonist of aryl hydrocarbon receptor (AhR)
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R2032982 |
CPI-455 |
CPI-455 is a specific, pan-KDM5 inhibitor with an IC50 of 10 nM for KDM5A.CPI-45
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R2032983 |
dasotraline |
Dasotraline is a triple reuptake inhibitor that blocks dopamine, norepinephrine,
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R2032984 |
DM1-Sme |
DM1-SMe is a potent maytansinoid microtubular inhibitor and an unconjugated DM1
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R2032985 |
MDK-5220 |
Orexin 2 Receptor Agonist is a potent (EC50 on OX2R is 23 nM) and OX2R-selective
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R2032986 |
Mitapivat |
Mitapivat is a pyruvate kinase isoenzyme M2 (PKM2) activator.
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R2032987 |
NVP-TNKS656 |
NVP-TNKS656 is a highly potent, selective, and orally active TNKS2 inhibitor wit
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R2032988 |
AZD0364 |
AZD-0364 is a potent and selective ERK2 inhibitor extracted from patent WO201708
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R2032989 |
E7820 |
E7820 is an angiogenesis inhibitor by suppressing integrin a2, a cell adhesion m
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R2032990 |
EPZ031686 |
EPZ031686 is an orally available SMYD3 inhibitor with an IC50 of 3 nM in cell-fr
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R2032991 |
LY3200882 |
LY3200882 is a novel and highly selective inhibitor of TGF-β receptor type 1 (TG
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R2032992 |
MK8617 |
MK-8617 is an orally active pan-inhibitor of hypoxia-inducible factor prolyl hyd
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R2032993 |
PF-3084014;Nirogacestat |
Nirogacestat (PF-3084014) is a reversible, noncompetitive, and selective γ-secre
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R2032994 |
PF9366 |
PF-9366 is a human methionine adenosyltransferase 2A (Mat2A) inhibitor, with an
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R2032995 |
Pyridostatin |
Pyridostatin is a G-quadruplexe stabilizer, with a Kd of 490 nM.
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R2032996 |
Ro25-6981 |
Ro 25-6981 is a potent and selective activity-dependent blocker of NMDA receptor
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R2032997 |
SC75741 |
SC75741 is a broad and efficient NF-κB inhibitor with an IC50 of 200 nM for p65.
|
R2032998 |
TP3654 |
TP-3654 is a second-generation Pim kinase inhibitor with Ki values of 5 and 42 n
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R2032999 |
AT406 hydrochloride |
AT-406 is a potent and orally bioavailable Smac mimetic and an antagonist of IAP
|
R2033000 |
BS194 |
BS194 is as a potent cyclin-dependent protein kinases (CDKs) inhibitor.
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R2033001 |
Cambinol |
Cambinol is a SIRT1 and SIRT2 inhibitor with IC50 values of 56 and 59 μM, respec
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R2033002 |
CCT241736 |
CCT241736 is a potent and orally bioavailable dual FLT3 and Aurora kinase inhibi
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R2033003 |
CFI-400437 |
CFI-400437 is potent against PLK4 (IC50 = 0.6 nM) and selective against other me
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