| R10988 |
XY1 NEW |
XY1 is a very close analogue of SGC707 (a potent, selective, and non-competitive
|
| R10989 |
SGC707 |
SGC707 is a potent, selective and cell-active allosteric inhibitor of protein ar
|
| R10990 |
SP2509 |
SP2509 is a selective histone demethylase LSD1 inhibitor with IC50 of 13 nM, sho
|
| R10992 |
IDO inhibitor 1 |
Epacadostat, also known as INCB024360 or INCB24360, is an orally available hydro
|
| R10994 |
ACT-678689 |
N/A
|
| R10996 |
Avitinib (AC0010) |
Avitinib (AC0010) is a pyrrolopyrimidine-based irreversible EGFR inhib
|
| R10997 |
GNF-7 |
GNF-7 is a potent type-II kinase Bcr-Abl inhibitor with IC50 of <5 nM, 61 nM,
|
| R10998 |
LY2608204 |
LY2608204 activates glucokinase (GK) with EC50 of 42 nM. Phase 2.
|
| R11000 |
Baricitinib phosphate;LY3009104 phosphate; INCB028050 phosphate |
Baricitinib (LY3009104, INCB028050) is a selective JAK1 and JAK2 inhibitor with
|
| R11001 |
LY2784544 |
Gandotinib (LY2784544) is a potent JAK2 inhibitor withIC50 of 3 n
|
| R11002 |
Abemaciclib; LY2835219 |
Abemaciclib (LY2835219) is a selective CDK4/6 inhibitor with IC50 values of 2 nM
|
| R11004 |
Micafungin;FK463 |
Micafungin (Mycamine; FK463) is an echinocandin antifungal drug which can inhibi
|
| R11006 |
Eliglustat (Synonyms: Genz 99067) |
Eliglustat (Tartrate) inhibits glucosylceramide synthase(GCS),thus reducing
|
| R11007 |
UK-2A |
N/A
|
| R11011 |
AM580 (Synonyms: CD336; NSC608001; Ro 40-6055) |
AM580 is a selective RARα agonist with IC50 and EC50 of 8 nM and 0.36 nM, respec
|
| R11012 |
Apixaban (BMS-562247-01) |
Apixaban is a highly selective, reversible inhibitor ofFactor Xa with
|
| R11013 |
Phenethyl caffeate |
Caffeic acid phenethyl ester is a potent and specific inhibitor of NF-κB&nb
|
| R11014 |
Brivaracetam;UCB 34714;UCB-34714;UCB34714; Briviact |
Brivaracetam has been tested in a comprehensive safety pharmacology, toxicology,
|
| R11015 |
Anamorelin ; RC-1291 |
Anamorelin(RC1291; ONO-7643) is a synthetic orally active ghrelin receptor agoni
|
| R11016 |
Rolapitant;SCH619734 |
Rolapitant (SCH619734) is a potent, selective and orally active neurokinin NK1 r
|
| R11017 |
Elbasvir;MK-8742 |
N/A
|
| R11018 |
Grazoprevir (MK-5172) |
Grazoprevir (MK-5172) is a selective inhibitor of Hepatitis C virus NS3/4a prote
|
| R11019 |
BMS863233; xl413 |
XL413 is a potent, selective and ATP competitive inhibitor of Cdc7, with an IC50
|
| R11021 |
1-NA-PP1 |
N/A
|
| R11023 |
ML-277 |
N/A
|