R2032873 |
BIX02565 |
BIX 02565 is a potent ribosomal S6 kinase 2 (RSK2) inhibitor with IC50 of 1.1 nM
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R2032874 |
CF-101;Piclidenoson |
Piclidenoson (IB-MECA; CF-101) is an agonist of the adenosine A3 receptor with E
|
R2032875 |
CPI-0610 |
CPI-0610 is a potent, selective, and cell-active BET inhibitor.CPI-0610 inhibits
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R2032876 |
GW0742 |
GW0742 is a potent PPARβ and PPARδ agonist, with an IC50 of 1 nM for human PPARδ
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R2032877 |
JD-5037 |
JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5
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R2032878 |
LTI-291 |
Gcase activator 1 is an activator of glucocerebrosidase (Gcase) extracted from p
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R2032879 |
MK8931;Verubecestat(MK-8931) |
Verubecestat (MK-8931) is a beta-secretase 1 (BACE1) inhibitor under investigati
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R2032880 |
PI-1840 |
PI-1840 is a potent and selective inhibitor for chymotrypsin-like (CT-L) (IC50 v
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R2032881 |
PNU74654 |
PNU-74654 is an inhibitor of Wnt/β-catenin pathway with an IC50 of 129.8 μM in N
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R2032882 |
RAD-140 |
RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen recepto
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R2032883 |
Rbin-1 |
Rbin-1 is a potent, reversible, and specific chemical inhibitor of eukaryotic ri
|
R2032884 |
SAR405 |
SAR405 is a first-in-class, selective, and ATP-competitive PI3K class III (PIK3C
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R2032885 |
VER49009 |
VER-49009 is a Hsp90 inhibitor, with an IC50 of 25 nM and a Kd of 78 nM.
|
R2032886 |
VER50589 |
VER-50589 is a Hsp90 inhibitor, with an IC50 of 21 nM and a Kd of 4.5 nM.
|
R2032887 |
AMG9810 |
AMG9810 is a selective and competitive vanilloid receptor 1 (TRPV1) antagonist w
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R2032888 |
TGR1202 |
Umbralisib (TGR-1202) is a novel PI3Kδ inhibitor, with IC50 and EC50 of 22.2 nM
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R2032889 |
Cenicriviroc |
Cenicriviroc is an orally active, dual CCR2/CCR5 antagonist, also inhibits both
|
R2032890 |
DiZPK |
DiZPK is a photocrosslinker for identifying direct protein-protein interactions
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R2032891 |
EED226 |
EED226 is a polycomb repressive complex 2 (PRC2) inhibitor, which binds to the K
|
R2032892 |
GLPG0187 |
GLPG0187 is a broad spectrum integrin receptor antagonist with antitumor activit
|
R2032893 |
ML385 |
ML385 is a specific nuclear factor erythroid 2-related factor 2 (NRF2) inhibitor
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R2032894 |
PF-06282999 |
PF-06282999 is a potent and selective myeloperoxidase inhibitor which is potenti
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R2032895 |
WT-161 |
WT-161 is a potent and selective HDAC6 inhibitor with an IC50 of 0.40 nM.
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R2032896 |
AP-III-a4 |
ENOblock(AP-III-a4) is a novel small molecule which is the first, nonsubstrate a
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R2032897 |
ARN272 |
ARN272 is an anandamide transport inhibitor.
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