| R2033083 |
AZD7507 |
AZD7507 is a potent and orally active CSF-1R inhibitor, with antitumor activity.
|
| R2033084 |
BB-Cl-Amidine |
BB-Cl-Amidine is a peptidylarginine deminase (PAD) inhibitor.
|
| R2033085 |
BTSA1 |
BTSA1 is a potent, high affinity and orally active BAX activator with an IC50 of
|
| R2033086 |
CVT-12012 |
CVT-12012 is a potent and orally bioavailable stearoyl-coA desaturase (SCD) inhi
|
| R2033087 |
Edicotinib(JNJ-40346527;JNJ-527) |
Edicotinib (JNJ-40346527; JNJ-527) is a potent, selective, brain penetrant and o
|
| R2033088 |
Gilteritinib |
Gilteritinib is a potent FLT3/AXL inhibitor with IC50s of 0.29 nM/0.73 nM, respe
|
| R2033089 |
JNJ42165279 |
JNJ-42165279 is a FAAH inhibitor with IC50 of 70 ± 8 nM and 313 ± 28 nM for hFAA
|
| R2033090 |
JNJ64619178 |
JNJ-64619178 is a selective, orally active and pseudo-irreversible PRMT5 inhibit
|
| R2033091 |
LKB1 |
Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/
|
| R2033092 |
LY2562175 |
LY2562175 is a potent and selective FXR agonist with an EC50 of 193 nM.
|
| R2033093 |
ML221 |
ML221 is a potent apelin (APJ) functional antagonist, inhibiting apelin-13-media
|
| R2033094 |
MRT67307 |
MRT67307 is a dual inhibitor of the IKKε and TBK-1 with IC50s of 160 and 19 nM,
|
| R2033095 |
PF-04418948 |
PF-04418948 is an orally active, potent and selective prostaglandin EP2 receptor
|
| R2033096 |
Pibrentasvir |
Pibrentasvir is a novel and pan-genotypic hepatitis C virus (HCV) NS5A inhibitor
|
| R2033097 |
RGX-104 |
RGX-104 is a small-molecule LXR agonist that modulates innate immunity via trans
|
| R2033098 |
SBI-0640756 |
SBI-0640756 (SBI-756) is a water soluble inhibitor of eIF4G1 and disrupts the eI
|
| R2033099 |
SM16 |
SM 16 is a ALK5/ALK4 kinase inhibitor with Kis of 10 and 1.5 nM, respectively.
|
| R2033100 |
Sotrastaurin |
Sotrastaurin is a potent and orally-active pan-PKC inhibitor, with Kis of 0.22 n
|
| R2033101 |
SP-13786 |
SP-13786 is a highly potent and selective inhibitor of fibroblast activation pro
|
| R2033102 |
SPHINX31 |
SPHINX31 is a potent and selective inhibitor of serine/arginine-rich protein kin
|
| R2033103 |
SR3677 |
SR-3677 is a potent and selective ROCK-II inhibitor with an IC50 of ~3 nM.
|
| R2033104 |
1358099-18-9 |
C25-140, a first-in-class, fairly selective TRAF6-Ubc13 inhibitor, directly bind
|
| R2033105 |
ACY775 |
ACY-775 is a potent and selective inhibitor of the of histone deacetylase 6 (HDA
|
| R2033106 |
Adavivint(SM04690;Lorecivivint) |
Adavivint (SM04690; Lorecivivint) is a potent and selective inhibitor of canonic
|
| R2033107 |
AR231453 |
AR 231453 is a potent, selective and orally available GPR119 agonist.
|