R2033079 |
NCGC00244536 |
NCGC00244536 is a potent KDM4B inhibitor with an IC50 of 10 nM.
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R2033080 |
INCB053914 phosphate |
INCB053914 phosphate is an inhibitor of Pim extracted from patent WO 2017044730
|
R2033081 |
SB297006 |
SB297006 is a CCR3 antagonist, which significantly inhibits proliferation and ne
|
R2033082 |
AMG176 |
AMG-176 is a potent, selective and orally bioavailable MCL-1 inhibitor, with a K
|
R2033083 |
AZD7507 |
AZD7507 is a potent and orally active CSF-1R inhibitor, with antitumor activity.
|
R2033084 |
BB-Cl-Amidine |
BB-Cl-Amidine is a peptidylarginine deminase (PAD) inhibitor.
|
R2033085 |
BTSA1 |
BTSA1 is a potent, high affinity and orally active BAX activator with an IC50 of
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R2033086 |
CVT-12012 |
CVT-12012 is a potent and orally bioavailable stearoyl-coA desaturase (SCD) inhi
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R2033087 |
Edicotinib(JNJ-40346527;JNJ-527) |
Edicotinib (JNJ-40346527; JNJ-527) is a potent, selective, brain penetrant and o
|
R2033088 |
Gilteritinib |
Gilteritinib is a potent FLT3/AXL inhibitor with IC50s of 0.29 nM/0.73 nM, respe
|
R2033089 |
JNJ42165279 |
JNJ-42165279 is a FAAH inhibitor with IC50 of 70 ± 8 nM and 313 ± 28 nM for hFAA
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R2033090 |
JNJ64619178 |
JNJ-64619178 is a selective, orally active and pseudo-irreversible PRMT5 inhibit
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R2033091 |
LKB1 |
Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/
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R2033092 |
LY2562175 |
LY2562175 is a potent and selective FXR agonist with an EC50 of 193 nM.
|
R2033093 |
ML221 |
ML221 is a potent apelin (APJ) functional antagonist, inhibiting apelin-13-media
|
R2033094 |
MRT67307 |
MRT67307 is a dual inhibitor of the IKKε and TBK-1 with IC50s of 160 and 19 nM,
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R2033095 |
PF-04418948 |
PF-04418948 is an orally active, potent and selective prostaglandin EP2 receptor
|
R2033096 |
Pibrentasvir |
Pibrentasvir is a novel and pan-genotypic hepatitis C virus (HCV) NS5A inhibitor
|
R2033097 |
RGX-104 |
RGX-104 is a small-molecule LXR agonist that modulates innate immunity via trans
|
R2033098 |
SBI-0640756 |
SBI-0640756 (SBI-756) is a water soluble inhibitor of eIF4G1 and disrupts the eI
|
R2033099 |
SM16 |
SM 16 is a ALK5/ALK4 kinase inhibitor with Kis of 10 and 1.5 nM, respectively.
|
R2033100 |
Sotrastaurin |
Sotrastaurin is a potent and orally-active pan-PKC inhibitor, with Kis of 0.22 n
|
R2033101 |
SP-13786 |
SP-13786 is a highly potent and selective inhibitor of fibroblast activation pro
|
R2033102 |
SPHINX31 |
SPHINX31 is a potent and selective inhibitor of serine/arginine-rich protein kin
|
R2033103 |
SR3677 |
SR-3677 is a potent and selective ROCK-II inhibitor with an IC50 of ~3 nM.
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