R2202001 |
Naringetol |
Naringenin is the predominant flavanone in grapefruit; displays strong anti-infl
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R2203201 |
NF-κΒ activator 2 |
NF-κΒ activator 2 is a potent and orally active NF-ҡB activator, with
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R2203202 |
Src Inhibitor 3 |
Src Inhibitor 3 is a potent, orally active c-terminal Src kinase (CSK) 
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R2203181 |
I-BET567 |
I-BET567 is a potent and orally active inhibitor of pan-BET candidate
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R2203222 |
Afn-1252 |
AFN-1252(Debio 1452) is a potent inhibitor of enoyl-acyl carrier protein reducta
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R2203212 |
MAX-40279 hydrochloride |
MAX-40279 hydrochloride is a dual and potent inhibitor of FLT3 kinase
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R2202111 |
GSK-2018682 |
GSK2018682 is an agonist for S1P1 and S1P5 receptor with pEC50s of 7.7 and 7.2,
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R2202112 |
PF3644022 |
PF-3644022 is a potent, selective, orally active and ATP-competitive MAPKAPK2 (M
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R2202113 |
SGC-SMARCA-BRDVIII |
SGC-SMARCA-BRDVIII is a potent and selective inhibitor of SMARCA2/4 and PB1(5),
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R2202114 |
BVT948 |
BVT948 is a protein tyrosine phosphatase (PTP) inhibitor which can also inhibit
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R2202115 |
PFI-90 |
PFI-90 is a selective inhibitor of histone demethylase (KDM3B) that inhibits PAX
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R2202116 |
TBAP-001 |
TBAP-001 (Synthesis 13), extracted from patent WO2015075483A1, is a pan-RAF kina
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R2202117 |
Robinetin |
Robinetin (3,3',4',5',7-Pentahydroxyflavone), a naturally occurring flavonoid wi
|
R2202118 |
MRTX1133 |
MRTX1133 is a noncovalent, potent, and selective KRAS G12D inhibitor. MRTX1133 o
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R2202119 |
HLY78 |
HLY78 is an activator of the Wnt/β-catenin signaling pathway, which targets the
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R2202120 |
SB-265610 |
SB-265610 is a selective, competitive, nonpeptide and allosteric CXCR2 antagonis
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R2202121 |
GSK2033 |
GSK2033 is a LXR antagonist with pIC50s of 7 and 7.4 for LXRα or LXRβ, respectiv
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R2202122 |
KL-11743 |
KL-11743 is a potent, orally active, and glucose-competitive inhibitor of the cl
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R2202123 |
Ch55 |
Ch55 is a potent synthetic retinoid. Ch55 binds to RAR-α and RAR-β receptors wit
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R2103226 |
Polyphyllin I |
Polyphyllin I is a bioactive constituent extracted from Paris polyphylla, h
|
R2001291 |
Coti-2 |
COTI-2, an anti-cancer drug with low toxicity, is an orally available third gene
|
R2204121 |
Lisavanbulin |
(S)-2,6-diamino-N-(4-(2-(2-(4-((2-cyanoethyl)amino)-1,2,5-oxadiazol-3-yl)-1H-ben
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R2204201 |
MRTX-1719 |
MRTX-1719 is a potent first-in-class selective inhibitor of the PRMT5/MTA&n
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R2202125 |
Remibrutinib(LOU064) |
Remibrutinib, is a potent and orally active bruton tyrosine kinase (BTK) inhibit
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R2202126 |
AZD9056 hydrochloride |
AZD9056 hydrochloride is a selective orally active inhibitor of P2X7 which plays
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