R2032252 |
Omipalisib;GSK2126458;GSK458 |
Omipalisib (GSK2126458) is a highly selective and potent inhibitor of PI3K with
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R2032253 |
GSK343 |
GSK343 is a highly potent and selective EZH2 inhibitor with an IC50 of 4 nM.
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R2032254 |
MK-0752 |
MK-0752 is a moderately potent γ-secretase inhibitor, which reduces Aβ40 product
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R2032255 |
Linsitinib(OSI906) |
Linsitinib (OSI-906) is a dual inhibitor of the IGF-1 receptor and IR with IC50s
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R2032256 |
Glasdegib(PF-04449913) |
Glasdegib (PF-04449913) is a potent and orally bioavailable smoothened inhibitor
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R2032257 |
Gedatolisib;PKI-587;PF-05212384 |
Gedatolisib (PKI-587) is a highly potent dual inhibitor of PI3Kα, PI3Kγ, and mTO
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R2032258 |
PD173074 |
PD173074 is a potent FGFR1 inhibitor with an IC50 of 25 nM and also inhibits VEG
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R2032259 |
PF573228 |
PF-573228 is a potent and selective FAK inhibitor with IC50 of 4 nM for purified
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R2032260 |
S1RA(E-52862) |
S1RA(E-52862) is a potent and selective sigma-1 receptor(σ1R, Ki=17 nM) antagoni
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R2032261 |
RO61-8048 |
Ro 61-8048 is a potent and selective inhibitor of kynurenine hydroxylase with IC
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R2032262 |
SB525334;SB-525334 |
SB 525334 is a potent and selective transforming growth factor β1 receptor (ALK5
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R2032263 |
TAK901 |
TAK-901 is a multi-targeted aurora inhibitor with IC50s of 21 and 15 nM for auro
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R2032264 |
Ricolinostat;ACY-1215;Rocilinostat |
Ricolinostat (ACY-1215) is a potent and selective HDAC6 inhibitor, with an IC50
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R2032265 |
TGR5 Receptor Agonist(CCDC) |
TGR5 Receptor Agonist (CCDC), a potent TGR5(GPCR19) agonist, shows improved pote
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R2032266 |
Orantinib(SU6668;TSU-68) |
Orantinib (SU6668; TSU-68) is a multi-targeted receptor tyrosine kinase inhibito
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R2032267 |
WP1066 |
WP1066 is an inhibitor of JAK2 and STAT3, and also shows effect on STAT5 and ERK
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R2032268 |
Mdivi-1 |
Mdivi-1 is a selective dynamin-related protein 1 (Drp1) inhibitor.Mdivi-1 is a m
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R2032269 |
SAR191801;hPGDS-IN-1 |
hPGDS-IN-1 is a hPGDS inhibitor ,with IC50 of 12 nM in the Fluorescence Polariza
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R2032270 |
GS967(GS-458967) |
GS967 (GS-458967) is a potent, and selective inhibitor of cardiac late sodium cu
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R2032271 |
ONO-4059 analog |
ONO-4059 analog is the analog of ONO-4059, ONO-4059 is a highly potent and selec
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R2032272 |
VRT-1353385;Sibofimloc(Antibiotic-202) |
Sibofimloc (Antibiotic-202) is an antibiotic compound, for treating bacterial in
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R2032273 |
ADX-47273 |
ADX-47273 is a positive allosteric modulator selective for the metabotropic glut
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R2032274 |
Ki16425(Debio0719) |
Ki16425 (Debio 0719) is a subtype-selective, competitive antagonist of the EDG-f
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R2032275 |
SAG |
SAG is a potent Smo receptor agonist which activates the Hedgehog signaling path
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R2032276 |
SB-242084 |
SB 242084 is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fo
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