R10915 |
GSK3235025;EPZ-015666;GSK-3235025 |
EPZ015666 is a potent, selective and orally bioavailable PRMT5 inhibitor with Ki
|
R10916 |
SKF-86002 |
SKF-86002 is a potent inhibitor of p38 MAP kinase wit IC50 of 0.5-1 uM; inhibits
|
R10917 |
Radotinib; IY-5511 |
Radotinib(IY-5511) is a novel and selective BCR-ABL1 tyrosine kinase inhibitor w
|
R10918 |
Liproxstatin-1 |
Liproxstatin-1 is a potent ferroptosis inhibitor.
|
R10919 |
Defactinib;VS-6063; PF-04554878 |
Defactinib (VS-6063; PF-04554878) is a novel FAK inhibitor with potential antian
|
R10920 |
HTH-01-015 |
HTH-01-015 is a potent and selective NUAK1 inhibitor with IC50 of 100 nM, >10
|
R10921 |
SD208 |
SD-208 is a selective TGF-βRI (ALK5) inhibitor with IC50 of 48 nM, >100-fold
|
R10925 |
ML324 |
ML324 is a selective inhibitor of jumonji histone demethylase (JMJD2) with IC50
|
R10926 |
ZK-811752; BX 471 |
BX471 (ZK-811752) is an orally active, potent and selective non-peptide CCR1 ant
|
R10927 |
Pilaralisib;SAR245408;XL147 |
Pilaralisib (XL147) is a selective and reversible class I PI3K inhibitor for PI3
|
R10929 |
UNC1215 |
UNC1215 is a potent and selective MBT (malignant brain tumor) antagonist, which
|
R10930 |
Icotinib |
Icotinib is a potent and specific EGFR inhibitor with IC50 of 5 nM, including th
|
R10931 |
Calcitriol; Vitamin D3 |
Calcitriol is the hormonally active form of vitamin D.
|
R10934 |
BI-847325 |
BI-847325 is an orally bioavailable, and selective dual MEK/Aurora kinase inhibi
|
R10935 |
AZD8186 |
N/A
|
R10936 |
FRAX597 |
FRAX597 is a potent, ATP-competitive inhibitor of group I PAKs with IC50 of 8 nM
|
R10937 |
AZD9496 |
AZD9496 is a potent and selective estrogen receptor (ERα) antagonist with an IC5
|
R10939 |
BMS-911543 |
BMS-911543 is a selective JAK2 inhibitor, with IC50s of 1.1 nM, less selective a
|
R10940 |
PRT-060318;PRT318 |
PRT-060318 (PRT318) is a novel selective inhibitor of the tyrosine kinase Syk wi
|
R10941 |
Alectinib(CH5424802; RO5424802; AF802) |
Alectinib (CH5424802) is a potent ALK inhibitor with IC50 of 1.9 nM in cell-free
|
R10942 |
Binimetinib; MEK162,ARRY-162,ARRY-438162 |
Binimetinib (MEK162, ARRY-162, ARRY-438162) is a potent inhibitor of MEK1/2 with
|
R10944 |
MK-801 ; Dizocilpine |
MK-801 (Dizocilpine) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist
|
R10946 |
Flibanserin;BIMT-17; BIMT-17BS |
Flibanserin (BIMT-17) is a full agonist of the serotonin 5-HT1A receptor (Ki=1 n
|
R10948 |
Lificiguat (YC-1) |
Lificiguat binds to the β subunit of soluble guanylyl cyclase(sGC) with Kd of 0.
|
R10950 |
ozanimod;RPC1063;RPC-1063 |
Ozanimod (RPC1063) is a selective oral S1P Receptor 1 modulator. Phase 3.
|